SCHEMBL6946320

SCHEMBL6946320

CCOC(=O)OC1CC(c2cccc(C(F)(F)F)c2)c2c(Cl)cc(Cl)cc2N1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
KMT2A Q03164 2/20 0.38
CACNA1F O60840 2/20 0.38
CACNA1D Q01668 2/20 0.38
CACNA1S Q13698 2/20 0.38
CACNA1C Q13936 2/20 0.38
PBRM1 Q86U86 1/20 0.38
POLB P06746 1/20 0.38
GUSB P08236 1/20 0.38
MAPT P10636 2/20 0.37
LMNA P02545 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HTT P42858 1/20 0.37
ACHE P22303 1/20 0.37
ELANE P08246 1/20 0.37
CYP2C9 P11712 1/20 0.37
MEN1 O00255 1/20 0.36
RECQL P46063 1/20 0.36
APOBEC3A P31941 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947977 0.89 MAPK1 (0.38) CACNA1FCACNA1DCACNA1SCACNA1CLMNA
SCHEMBL6944762 0.88 ALDH1A1 (0.37) ALDH1A1KMT2ALMNAACHE
SCHEMBL6951129 0.87 MEN1 (0.39) KMT2AMEN1
SCHEMBL6949316 0.86 ALDH1A1 (0.35) ALDH1A1
SCHEMBL6770056 0.85 PBRM1 (0.41) ALDH1A1KMT2ACACNA1FCACNA1DCACNA1S
SCHEMBL7546562 0.84 ABCC1 (0.38) ALDH1A1LMNAHTT
SCHEMBL7489535 0.83 CYP2D6 (0.36) CYP2C9
SCHEMBL6952784 0.83 GAA (0.35)
SCHEMBL6945541 0.83 MAPK1 (0.35)
SCHEMBL6946334 0.83 MMP13 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003522758-A 2003-07-29 JP claimed
EP-1254118-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2002-11-06 EP claimed
WO-2001058875-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2001-08-16 WO claimed
EP-1254118-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2002-11-06 EP disclosed
WO-2001058875-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2001-08-16 WO disclosed