SCHEMBL6946443

SCHEMBL6946443

NS(=O)(=O)c1ccc(CC(Cc2ccc(OP(=O)(O)C(F)F)cc2)(C(=O)c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.53
CA12 O43570 14/20 0.44
CA1 P00915 14/20 0.44
CA2 P00918 14/20 0.44
CA4 P22748 14/20 0.44
CA5A P35218 14/20 0.44
CA7 P43166 14/20 0.44
CA9 Q16790 14/20 0.44
CA5B Q9Y2D0 14/20 0.44
PTPRC P08575 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6948321 0.90 PTPN1 (0.61) PTPN1PTPRC
SCHEMBL7884360 0.85 PTPN1 (0.75) PTPN1PTPRC
SCHEMBL6946012 0.81 PTPN1 (0.80) PTPN1PTPRC
SCHEMBL7161145 0.80 PTPN1 (0.69) PTPN1PTPRC
SCHEMBL7888262 0.78 PTPN1 (0.56) PTPN1CA12CA1CA2CA4
SCHEMBL6944056 0.77 PTPN1 (0.62) PTPN1PTPRC
SCHEMBL7165297 0.77 PTPN1 (0.54) PTPN1PTPRC
SCHEMBL6946043 0.77 CA2 (0.45) CA12CA1CA2CA4CA5A
SCHEMBL6948696 0.77 PTPN1 (0.61) PTPN1PTPRC
SCHEMBL6951395 0.77 PTPN1 (0.51) PTPN1CA12CA1CA2CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115729-B1 PHOSPHONIC ACID DERIVATIVES AS INHIBITORS OF PTP-1B MERCK FROSST CANADA INC (CA) 2003-02-19 EP disclosed
US-6174874-B1 ANTIDIABETIC,-CARCINOGENIC AGENTS; IMPROVING GLUCOSE TOLERANCE/INSULIN-SENSITIVITY; PREVENTING/TREATING OBESITY AND NEURODEGENERATIVE DISEASES; E.G. 1,3-BIS-((PHOSPHONODI-FLUOROMETHYL)PHENYL)-2-DICARBOXYPROPANE MERCK FROSST CANADA & CO. (CA) 2001-01-16 US disclosed