SCHEMBL6947000

SCHEMBL6947000

CS(=O)(=O)OCCC[C@H](NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 2/20 0.53
SIRT1 Q96EB6 2/20 0.53
CTSL P07711 2/20 0.52
CTSS P25774 2/20 0.52
FOLH1 Q04609 2/20 0.51
ITGB3 P05106 8/20 0.49
ITGA2B P08514 6/20 0.49
ITGAV P06756 2/20 0.48
TGM2 P21980 1/20 0.48
MMP2 P08253 1/20 0.48
MMP9 P14780 1/20 0.48
CTSK P43235 3/20 0.48
MME P08473 1/20 0.48
ECE1 P42892 1/20 0.48
CTSB P07858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8671689 1.00 SIRT2 (0.53) SIRT2SIRT1CTSLCTSSFOLH1
SCHEMBL26641013 0.96 SIRT2 (0.55) SIRT2SIRT1CTSLCTSSFOLH1
SCHEMBL26641008 0.96 SIRT2 (0.55) SIRT2SIRT1CTSLCTSSFOLH1
SCHEMBL28723314 0.93 CTSK (0.50) SIRT2SIRT1CTSLCTSSFOLH1
SCHEMBL28723315 0.93 CTSK (0.50) SIRT2SIRT1CTSLCTSSFOLH1
SCHEMBL9301974 0.88 SYK (0.52) SIRT2SIRT1CTSLCTSSITGB3
SCHEMBL4972916 0.85 CTSK (0.52) CTSLCTSSITGB3ITGA2BCTSK
SCHEMBL4972907 0.85 CTSK (0.52) CTSLCTSSITGB3ITGA2BCTSK
SCHEMBL5141850 0.85 CTRB1 (0.49) CTSLCTSSCTSKCTSB
SCHEMBL5141853 0.85 CTRB1 (0.49) CTSLCTSSCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0758328-B1 ANTI-CANCER COMPOUNDS CONTAINING CYCLOPENTAQUINAZOLINE RING BTG INT LTD (GB) 2003-07-16 EP disclosed
US-5747499-A CYCLOPENTAQUINAZOLINE COMPOUNDS CYCLOPENTAQUINAZOLINE COMPOUNDS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1998-05-05 US disclosed
EP-0758328-A1 ANTI-CANCER COMPOUNDS CONTAINING CYCLOPENTAQUINAZOLINE RING BTG INTERNATIONAL LIMITED (GB) 1997-02-19 EP disclosed
WO-1995030673-A1 ANTI-CANCER COMPOUNDS CONTAINING CYCLOPENTAQUINAZOLINE RING BRITISH TECHNOLOGY GROUP LIMITED (GB) 1995-11-16 WO disclosed