SCHEMBL6947033

SCHEMBL6947033

N#C[C@@H](CCC(=O)O)NC(=O)OCc1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.53
CTSL P07711 11/20 0.53
CTSS P25774 11/20 0.53
CTSK P43235 8/20 0.53
CTSB P07858 3/20 0.52
HTT P42858 1/20 0.51
FOLH1 Q04609 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11660684 0.88 HTT (0.52) TACR1CTSLCTSSCTSKCTSB
SCHEMBL10556998 0.88 HTT (0.52) TACR1CTSLCTSSCTSKCTSB
SCHEMBL24853554 0.86 CTSS (0.60) TACR1CTSLCTSSCTSKCTSB
SCHEMBL29249016 0.86 CTSS (0.60) TACR1CTSLCTSSCTSKCTSB
SCHEMBL8728480 0.86 CTSL (0.52) TACR1CTSLCTSSCTSKCTSB
SCHEMBL7418478 0.86 TACR1 (0.55) TACR1CTSLCTSSCTSKCTSB
SCHEMBL6312394 0.85 CTSL (0.65) TACR1CTSLCTSSCTSKCTSB
SCHEMBL6318841 0.85 CTSL (0.65) TACR1CTSLCTSSCTSKCTSB
SCHEMBL392814 0.85 CTSL (0.65) TACR1CTSLCTSSCTSKCTSB
SCHEMBL16357709 0.84 CTSS (0.67) TACR1CTSLCTSSCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0758328-B1 ANTI-CANCER COMPOUNDS CONTAINING CYCLOPENTAQUINAZOLINE RING BTG INT LTD (GB) 2003-07-16 EP disclosed
US-5747499-A CYCLOPENTAQUINAZOLINE COMPOUNDS CYCLOPENTAQUINAZOLINE COMPOUNDS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1998-05-05 US disclosed
EP-0758328-A1 ANTI-CANCER COMPOUNDS CONTAINING CYCLOPENTAQUINAZOLINE RING BTG INTERNATIONAL LIMITED (GB) 1997-02-19 EP disclosed
WO-1995030673-A1 ANTI-CANCER COMPOUNDS CONTAINING CYCLOPENTAQUINAZOLINE RING BRITISH TECHNOLOGY GROUP LIMITED (GB) 1995-11-16 WO disclosed