SCHEMBL6947089

SCHEMBL6947089

COc1c(CN(C)C)cc(Cc2ccccc2)cc1C(=O)CC(=O)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 6/20 0.40
PTPN2 P17706 1/20 0.40
PTPN6 P29350 1/20 0.40
ERCC5 P28715 5/20 0.40
FEN1 P39748 5/20 0.40
CNR1 P21554 2/20 0.38
CNR2 P34972 2/20 0.38
MMP1 P03956 1/20 0.37
MMP9 P14780 1/20 0.37
MMP13 P45452 1/20 0.37
ADAM17 P78536 1/20 0.37
MTNR1A P48039 1/20 0.37
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947887 0.88 PTPN1 (0.38) PTPN1PTPN2PTPN6ERCC5FEN1
SCHEMBL6947937 0.87 PTPN1 (0.43) PTPN1PTPN2PTPN6ERCC5FEN1
SCHEMBL6944964 0.84 ALDH1A1 (0.46) PTPN1PTPN2PTPN6CNR1CNR2
SCHEMBL6947888 0.84 ERCC5 (0.42) PTPN1PTPN2PTPN6ERCC5FEN1
SCHEMBL6946973 0.82 KDM4E (0.46) PTPN1ERCC5FEN1ALDH1A1MEN1
Dimethylamine SCHEMBL6947095 0.81 ERCC5 (0.50) PTPN1ERCC5FEN1CNR1CNR2
SCHEMBL6943825 0.81 ERCC5 (0.43) PTPN1PTPN2PTPN6ERCC5FEN1
SCHEMBL6947664 0.79 MEN1 (0.43) ALDH1A1MEN1KMT2AKDM4E
SCHEMBL6949373 0.78 ERCC5 (0.49) PTPN1ERCC5FEN1CNR1CNR2
SCHEMBL6943490 0.78 ALDH1A1 (0.45) ALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed