SCHEMBL6944964

SCHEMBL6944964

COc1c(CN(C)C)cc(Cc2ccccc2)cc1C(C)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PTPN1 P18031 3/20 0.45
PTPN2 P17706 1/20 0.45
PTPN6 P29350 1/20 0.45
LMNA P02545 1/20 0.44
MTNR1A P48039 2/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
CNR1 P21554 2/20 0.39
CNR2 P34972 2/20 0.39
MAPK1 P28482 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HNF4A P41235 1/20 0.38
MTNR1B P49286 1/20 0.37
TSHR P16473 2/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947089 0.84 PTPN1 (0.40) ALDH1A1MEN1KMT2APTPN1PTPN2
SCHEMBL6951260 0.80 TUBB4A (0.47) ALDH1A1MEN1KMT2APTPN1PTPN2
SCHEMBL6949776 0.79 ALDH1A1 (0.41) ALDH1A1MEN1KMT2ALMNASLC6A2
SCHEMBL9192926 0.77 PTPN1 (0.61) ALDH1A1PTPN1PTPN2PTPN6LMNA
SCHEMBL7077211 0.76 SMN1; SMN2 (0.46) ALDH1A1MEN1KMT2ALMNAMAPK1
SCHEMBL6947887 0.75 PTPN1 (0.38) ALDH1A1PTPN1PTPN2PTPN6LMNA
Zinc Ion SCHEMBL9192923 0.75 PTPN1 (0.51) ALDH1A1PTPN1PTPN2PTPN6LMNA
SCHEMBL6949242 0.73 LMNA (0.42) ALDH1A1MEN1KMT2APTPN1PTPN2
SCHEMBL2097755 0.70 LTA4H (0.53) PTPN1PTPN2PTPN6LMNACNR1
SCHEMBL6947937 0.70 PTPN1 (0.43) PTPN1PTPN2PTPN6MTNR1ACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed