SCHEMBL6943490

SCHEMBL6943490

COc1cc(Cc2ccccc2)cc(C(=O)CC(=O)C(=O)O)c1OCCCN(C)C

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
HRH1 P35367 3/20 0.44
LTA4H P09960 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
KDM4E B2RXH2 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
THRA P10827 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6951319 0.87 ERCC5 (0.39) ALDH1A1KMT2AKDM4ESMN1; SMN2
Dimethylamine SCHEMBL6943493 0.86 LMNA (0.42) ALDH1A1KMT2AKDM4ESMN1; SMN2
SCHEMBL6946187 0.85 PTPN1 (0.47) ALDH1A1MEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL6946973 0.85 KDM4E (0.46) ALDH1A1MEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL6951986 0.84 KDM4E (0.37) ALDH1A1MEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL6949341 0.80 KDM4E (0.52) ALDH1A1HRH1LTA4HKDM4ESMN1; SMN2
SCHEMBL6948187 0.80 ERCC5 (0.40) ALDH1A1MEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL6951318 0.79 ERCC5 (0.39) ALDH1A1MEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL6947089 0.78 PTPN1 (0.40) ALDH1A1MEN1KMT2AKDM4E
SCHEMBL6947620 0.78 LTA4H (0.50) ALDH1A1HRH1LTA4HKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP claimed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP claimed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed