SCHEMBL6947183

SCHEMBL6947183

COc1ccc(CC(/C=C/c2ccccc2)([C@H](C(=O)NOC2CCCCO2)[C@@H](CC(C)C)C(=O)NN)S(C)(=O)=O)cc1

nearest known ligand 0.32

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KLK7 P49862 1/20 0.32
MMP1 P03956 8/20 0.31
MMP13 P45452 4/20 0.31
MMP2 P08253 2/20 0.31
MMP3 P08254 2/20 0.31
MMP8 P22894 1/20 0.31
MMP9 P14780 3/20 0.30
CTSD P07339 1/20 0.30
BACE1 P56817 1/20 0.30
BACE2 Q9Y5Z0 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MAPK1 P28482 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
PLA2G2A P14555 1/20 0.30
CTSK P43235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6943971 0.94 ADAM17 (0.32) MMP2MMP3MMP9
SCHEMBL6945328 0.92 ADAM17 (0.33) MMP2MMP9
SCHEMBL6943358 0.89 ADAM17 (0.32) ALDH1A1MMP2MMP9
SCHEMBL6942209 0.89 ADAM17 (0.33) ALDH1A1MMP2MMP9
SCHEMBL8111706 0.89 ADAM17 (0.33) ALDH1A1MMP2MMP9
SCHEMBL6943556 0.89 ADAM17 (0.33) ALDH1A1MMP2MMP9
SCHEMBL6944327 0.88 TGFBR1 (0.31)
SCHEMBL6946835 0.88 ADAM17 (0.32) MMP2MMP9
SCHEMBL6940018 0.88 MMP2 (0.33) ALDH1A1KLK7MMP1MMP13MMP2
SCHEMBL6946731 0.87 ADAM17 (0.33) MMP1MMP2MMP3MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed
EP-0993442-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-04-19 EP disclosed
WO-1999001428-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-01-14 WO disclosed