SCHEMBL6947723

SCHEMBL6947723

O=C(O)c1ccc2[nH]cc(CCCCN3CCCC(Cc4ccccc4)C3)c2c1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.58
ALOX15 P16050 1/20 0.58
APEX1 P27695 1/20 0.58
KMT2A Q03164 1/20 0.58
HSD17B10 Q99714 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
HTR1A P08908 8/20 0.52
HTR1D P28221 1/20 0.51
HTR1B P28222 1/20 0.51
SLC6A4 P31645 5/20 0.51
ACHE P22303 1/20 0.49
SLC6A2 P23975 1/20 0.49
SLC6A3 Q01959 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959565 0.91 HTR1A (0.63) KDM4EALOX15APEX1KMT2AHSD17B10
SCHEMBL27318120 0.89 KDM4E (0.57) KDM4EALOX15APEX1KMT2AHSD17B10
SCHEMBL7356374 0.87 HTR1A (0.51) HTR1AHTR1DHTR1BSLC6A4
SCHEMBL6958552 0.86 MPO (0.61) HTR1AHTR1DHTR1BSLC6A4
SCHEMBL7358948 0.86 HTR1A (0.54) KMT2AHTR1AHTR1DHTR1BSLC6A4
SCHEMBL6957729 0.86 MPO (0.61) HTR1AHTR1DHTR1BSLC6A4
SCHEMBL6951363 0.86 HTR1A (0.55) KMT2ATDP1HTR1AHTR1DHTR1B
SCHEMBL6952634 0.86 MPO (0.61) HTR1AHTR1DHTR1BSLC6A4
SCHEMBL6950516 0.86 HTR1A (0.56) HTR1AHTR1DHTR1BSLC6A4
SCHEMBL7879034 0.84 HTR1A (0.55) HTR1AHTR1DHTR1BSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP claimed
US-6333339-B1 CENTRAL SYSTEM DISORDERS, SCHIZOPHRENIA AND COGNITION ACTIVATORS MERCK PATENT GELLSCHAFT MIT BESCHRANKTER (DE) 2001-12-25 US claimed
EP-0993458-A1 3-BENZYLPIPERIDINE MERCK PATENT GmbH (DE) 2000-04-19 EP claimed
WO-1998057953-A1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 1998-12-23 WO claimed
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP disclosed
US-6333339-B1 CENTRAL SYSTEM DISORDERS, SCHIZOPHRENIA AND COGNITION ACTIVATORS MERCK PATENT GELLSCHAFT MIT BESCHRANKTER (DE) 2001-12-25 US disclosed
EP-0993458-A1 3-BENZYLPIPERIDINE MERCK PATENT GmbH (DE) 2000-04-19 EP disclosed
WO-1998057953-A1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 1998-12-23 WO disclosed