SCHEMBL6948825

SCHEMBL6948825

C=C(c1ccccc1)n1c(=O)n(CC)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ATM Q13315 1/20 0.46
TMEM97 Q5BJF2 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
HTR3A P46098 1/20 0.44
HTR4 Q13639 1/20 0.44
PGR P06401 1/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 1/20 0.43
APEX1 P27695 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6951613 0.88 PGR (0.46) MEN1KMT2AATMPGRSLC6A2
SCHEMBL8119434 0.83 ALDH1A1 (0.46) ALDH1A1
SCHEMBL6644290 0.82 MEN1 (0.41) MEN1KMT2AATMAPEX1ALDH1A1
SCHEMBL8565489 0.82 MEN1 (0.44) MEN1KMT2AATMAPEX1GAA
SCHEMBL3301756 0.80 TMEM97 (0.51) MEN1KMT2ATMEM97SIGMAR1HTR3A
SCHEMBL6947807 0.79 ALDH1A1 (0.47) PGRSLC6A2ALDH1A1
SCHEMBL6582840 0.76 TMEM97 (0.53) MEN1KMT2ATMEM97SIGMAR1HTR3A
SCHEMBL6588314 0.76 TMEM97 (0.50) MEN1KMT2ATMEM97SIGMAR1HTR3A
SCHEMBL4621924 0.75 ALDH1A1 (0.59) MEN1KMT2APGRSLC6A2SLC6A4
SCHEMBL6945702 0.71 SLC6A2 (0.42) HTR4SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1105388-B1 N-SUBSTITUTED AZABICYCLOHEPTANE DERIVATIVES, PRODUCTION AND USE THEREOF BASF AG (DE) 2003-05-02 EP disclosed
US-6458821-B1 THE NOVEL SUBSTANCES ARE SUITABLE FOR CONTROLLING DISEASES. INTERESTING PROPERTIES AS POTENTIAL NEUROLEPTICS AND ANTIDEPRESSANTS ABBOTT LABORATORIES 2002-10-01 US disclosed