SCHEMBL6948894

SCHEMBL6948894

COc1ccc(C(=O)Nc2ccncc2)c2cc(C(C)C)oc12

nearest known ligand 0.74

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 11/20 0.74
PDE4B Q07343 11/20 0.74
PDE4C Q08493 11/20 0.74
PDE4D Q08499 11/20 0.74
KCNMA1 Q12791 1/20 0.54
MAPK1 P28482 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MEN1 O00255 1/20 0.51
ALDH1A1 P00352 1/20 0.51
PKM P14618 1/20 0.51
KMT2A Q03164 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
JAK2 O60674 2/20 0.49
TYK2 P29597 1/20 0.48
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5722732 0.84 PDE4A (0.74) PDE4APDE4BPDE4CPDE4DKCNMA1
SCHEMBL7643622 0.83 PDE4A (0.60) PDE4APDE4BPDE4CPDE4D
SCHEMBL6950329 0.81 PDE4D (0.88) PDE4APDE4BPDE4CPDE4D
SCHEMBL7909583 0.81 PDE4A (0.70) PDE4APDE4BPDE4CPDE4DKCNMA1
SCHEMBL5722709 0.79 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DKCNMA1
SCHEMBL6954572 0.78 PDE4D (0.50) PDE4APDE4BPDE4CPDE4DMAPK1
SCHEMBL5023240 0.76 PDE4B (0.63) PDE4APDE4BPDE4CPDE4DKCNMA1
SCHEMBL6950936 0.76 PDE4D (0.67) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL5017990 0.76 PDE4D (0.62) PDE4APDE4BPDE4CPDE4DKCNMA1
SCHEMBL7916544 0.76 PDE4D (0.67) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923568-B9 NOVEL BENZOFURAN-4-CARBOXAMIDES ALTANA PHARMA AG (DE) 2003-08-13 EP disclosed
EP-0923568-B1 NOVEL BENZOFURAN-4-CARBOXAMIDES ALTANA PHARMA AG (DE) 2002-12-11 EP disclosed
US-6211203-B1 RESPIRATORY SYSTEM DISORDERS, ANTIINFLAMMATORY AGENTS, ENZYME INHIBITORS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2001-04-03 US disclosed
EP-0923568-A1 NOVEL BENZOFURAN-4-CARBOXAMIDES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1999-06-23 EP disclosed
WO-1998007715-A9 NOVEL BENZOFURAN-4-CARBOXAMIDES BYK GULDEN LOMBERG CHEM FAB (DE) 1999-04-29 WO disclosed
WO-1998007715-A1 NOVEL BENZOFURAN-4-CARBOXAMIDES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-02-26 WO disclosed