SCHEMBL6949341

SCHEMBL6949341

CC(C)Oc1c(OCCN(C)C)cc(Cc2ccccc2)cc1C(=O)CC(=O)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.52
ALDH1A1 P00352 6/20 0.52
HRH1 P35367 3/20 0.43
DRD2 P14416 1/20 0.42
DRD1 P21728 1/20 0.42
DRD4 P21917 1/20 0.42
DRD5 P21918 1/20 0.42
LMNA P02545 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
BRPF1 P55201 1/20 0.41
LTA4H P09960 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
MCHR1 Q99705 3/20 0.40
THRA P10827 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6951272 0.86 KDM4E (0.43) KDM4EALDH1A1LMNATDP1
Dimethylamine SCHEMBL6949345 0.86 SMN1; SMN2 (0.41) KDM4EALDH1A1LMNATDP1SMN1; SMN2
SCHEMBL6948187 0.84 ERCC5 (0.40) KDM4EALDH1A1LMNATDP1SMN1; SMN2
SCHEMBL6947620 0.82 LTA4H (0.50) KDM4EALDH1A1HRH1DRD2DRD1
SCHEMBL6947887 0.82 PTPN1 (0.38) KDM4EALDH1A1LMNATDP1
SCHEMBL6950058 0.81 ERCC5 (0.39) KDM4EALDH1A1LMNATDP1
SCHEMBL6943490 0.80 ALDH1A1 (0.45) KDM4EALDH1A1HRH1LTA4HSMN1; SMN2
SCHEMBL6947879 0.79 ERCC5 (0.41) KDM4ELMNATDP1
SCHEMBL6951318 0.77 ERCC5 (0.39) KDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL5148099 0.75 IDO1 (0.44) KDM4EALDH1A1LMNATDP1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US claimed
EP-1082121-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-02-05 EP disclosed
US-6380249-B1 HIV integrase inhibitors MERCK & CO., INC. 2002-04-30 US disclosed
EP-1082121-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-14 EP disclosed
WO-1999062520-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed