SCHEMBL6950

SCHEMBL6950

Cc1noc(-c2ccc(Br)cc2)c1-c1ccc(I)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 5/20 0.39
BRD2 P25440 1/20 0.39
TDO2 P48775 1/20 0.37
ALOX5AP P20292 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
IKBKB O14920 1/20 0.35
CHUK O15111 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
LMNA P02545 1/20 0.34
MLYCD O95822 1/20 0.34
EDNRB P24530 2/20 0.33
EDNRA P25101 2/20 0.33
HTT P42858 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6511644 0.85 BRD4 (0.56) BRD4BRD2TDO2ALOX5APEDNRB
SCHEMBL6514108 0.81 ALDH1A1 (0.40) BRD4BRD2TDO2ALOX5APMEN1
SCHEMBL11929 0.81 BRD4 (0.34) BRD4ALOX5APMEN1KMT2ATRPV1
SCHEMBL18597730 0.80 MEN1 (0.39) MEN1KMT2ATRPV1LMNAEDNRB
SCHEMBL6513072 0.79 PTGS2 (0.56) EDNRBEDNRACYP1A2CYP3A4CYP2C9
SCHEMBL6517910 0.78 CA2 (0.54) LMNAEDNRBEDNRACYP1A2CYP3A4
SCHEMBL1772573 0.75 BRD4 (0.66) BRD4BRD2MEN1KMT2ALMNA
SCHEMBL27886960 0.75 EDNRB (0.45) MEN1KMT2ATRPV1EDNRBEDNRA
SCHEMBL21105338 0.73 BRD4 (0.68) BRD4BRD2TDO2ALOX5APPTGS2
SCHEMBL25406124 0.73 MEN1 (0.39) BRD4BRD2MEN1KMT2ATRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483252-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041694-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed