SCHEMBL6950164

SCHEMBL6950164

CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)CC(O)c1cccc2[nH]c(CCc3ccccc3)nc12

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.47
PARP1 P09874 1/20 0.43
PARP3 Q9Y6F1 1/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PTGS2 P35354 1/20 0.41
PIN1 Q13526 2/20 0.41
POLB P06746 3/20 0.40
ELANE P08246 1/20 0.40
RAB9A P51151 1/20 0.39
MMP2 P08253 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
MMP13 P45452 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6943129 1.00 TP53 (0.47) TP53PARP1PARP3ALDH1A1MEN1
SCHEMBL29828622 0.84 CHEK1 (0.48) ALDH1A1RAB9AMMP2
SCHEMBL6945277 0.84 CHEK1 (0.48) ALDH1A1RAB9AMMP2
SCHEMBL6953837 0.84 CHEK1 (0.43) ALDH1A1POLBRAB9AMMP2RXFP1
SCHEMBL6945574 0.81 CHEK1 (0.46) ALDH1A1KMT2ARAB9AMMP2
SCHEMBL6952443 0.80 BRD4 (0.46) PARP1ALDH1A1RAB9AMMP2
SCHEMBL7653156 0.79 ALDH1A1 (0.42) PARP1ALDH1A1RAB9AMMP2
SCHEMBL529009 0.79 RAB9A (0.48) ALDH1A1RAB9A
SCHEMBL6950391 0.77 CHEK1 (0.52) PARP1ALDH1A1RAB9AMMP2
SCHEMBL7654820 0.77 ALDH1A1 (0.50) ALDH1A1MEN1KMT2APOLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0936218-B1 BENZIMIDAZOLE DERIVATIVES MOCHIDA PHARM CO LTD (JP) 2003-04-02 EP disclosed
US-6387938-B1 Benzimidazole derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2002-05-14 US disclosed
EP-0936218-A1 NOVEL BENZIMIDAZOLE DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1999-08-18 EP disclosed