SCHEMBL6950169

SCHEMBL6950169

CC(=O)OCc1ccc(C(=O)O)cc1[N+](=O)[O-]

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.55
TSHR P16473 2/20 0.55
HCAR3 P49019 12/20 0.51
LMNA P02545 1/20 0.51
APEX1 P27695 1/20 0.48
PDK1 Q15118 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7109468 0.90 ALDH1A1 (0.54) TSHRLMNAPDK1
SCHEMBL27548058 0.89 CASP6 (0.55) CASP6TSHRHCAR3LMNA
SCHEMBL27544736 0.86 PDK1 (0.49) HCAR3LMNAPDK1
SCHEMBL4175596 0.85 CASP6 (0.58) CASP6TSHRHCAR3LMNAAPEX1
SCHEMBL17053413 0.85 PDK1 (0.45) TSHRHCAR3LMNAPDK1
SCHEMBL14714240 0.84 KMT2A (0.42) LMNAPDK1
SCHEMBL13264670 0.83 CASP6 (0.55) CASP6TSHRHCAR3LMNAAPEX1
SCHEMBL6886014 0.83 ALDH1A1 (0.46) LMNAPDK1
SCHEMBL19193928 0.82 TSHR (0.50) TSHRLMNA
SCHEMBL27736701 0.82 CYP1A2 (0.59) TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0751765-B1 SULFONAMIDE DERIVATIVES AND THEIR USE PHARMACOPEIA INC (US) 2003-05-07 EP disclosed
EP-0766826-B1 SYNTHESIS OF COMBINATORIAL LIBRARIES PHARMACOPEIA INC (US) 2002-05-22 EP disclosed
US-5756810-A Process of preparing 3-nitro benzoate compounds in lower alkanol PHARMACOPEIA, INC. (US) 1998-05-26 US disclosed
EP-0766826-A4 SYNTHESIS OF COMBINATORIAL LIBRARIES PHARMACOPEIA INC (US) 1998-02-11 EP disclosed
US-5663046-A DIRECTLY DIVIDING THE CONTENTS OF EACH SUB-POOL INTO THE SUB-POOLS FOR THE NEXT STEP IN THE SYNTHETIC SCHEME REDUCES THE CALCULABLE ERROR FROM THE THAT OF SPLIT SYNTHESIS PHARMACOPEIA, INC. (US) 1997-09-02 US disclosed
EP-0751765-A4 SULFONAMIDE DERIVATIVES AND THEIR USE PHARMACOPEIA INC (US) 1997-05-28 EP disclosed
EP-0766826-A1 SYNTHESIS OF COMBINATORIAL LIBRARIES PHARMACOPEIA, INC. (US) 1997-04-09 EP disclosed
US-5618825-A ENZYME INHIBITORS; ANTICOAGULANTS; VISION DISORDERS PHARMACOPEIA, INC. (US) 1997-04-08 US disclosed
EP-0751765-A1 SULFONAMIDE DERIVATIVES AND THEIR USE PHARMACOPEIA, INC. (US) 1997-01-08 EP disclosed
WO-1995035503-A1 SYNTHESIS OF COMBINATORIAL LIBRARIES PHARMACOPEIA, INC. (US) 1995-12-28 WO disclosed
WO-1995024186-A1 SULFONAMIDE DERIVATIVES AND THEIR USE PHARMACOPEIA, INC. (US) 1995-09-14 WO disclosed