SCHEMBL6950805

SCHEMBL6950805

CC(C)(C)OC(=O)N[C@@H](Cc1cncn1C(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.50
ITGA4 P13612 2/20 0.44
ITGB7 P26010 2/20 0.44
ITGB3 P05106 2/20 0.43
ITGA2B P08514 2/20 0.43
MAPK1 P28482 1/20 0.43
PPARA Q07869 6/20 0.41
PPARG P37231 5/20 0.41
PTPN1 P18031 2/20 0.40
PPARD Q03181 2/20 0.39
SCN9A Q15858 1/20 0.39
CTSS P25774 3/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CTSK P43235 1/20 0.39
ITGB1 P05556 1/20 0.39
ITGAV P06756 1/20 0.39
ITGB5 P18084 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957298 1.00 ACE (0.50) ACEITGA4ITGB7ITGB3ITGA2B
SCHEMBL22403247 0.91 ACE (0.40) ACEITGA4ITGB7CTSSCTSL
SCHEMBL16819882 0.88 ACE (0.47) ACEITGA4ITGB7ITGB3ITGA2B
SCHEMBL15426849 0.88 ACE (0.47) ACEITGA4ITGB7ITGB3ITGA2B
SCHEMBL8054432 0.88 CTSS (0.40) ACECTSSCTSLCTSBCTSK
SCHEMBL3007905 0.85 ACE (0.49) ACEITGA4ITGB7ITGB3ITGA2B
SCHEMBL7052233 0.85 ACE (0.49) ACEITGA4ITGB7ITGB3ITGA2B
SCHEMBL3007900 0.85 ACE (0.49) ACEITGA4ITGB7ITGB3ITGA2B
SCHEMBL15412931 0.85 MEN1 (0.43) ACE
SCHEMBL13811785 0.84 ACE (0.36) ACEITGA4ITGB7CTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9085587-B2 Inhibitors of hepatitis C virus PRESIDIO PHARMACEUTICALS, INC. (US) 2015-07-21 US disclosed
EP-0757677-B1 BENZOCYCLOHEXYLIMIDAZOLETHIONE DERIVATIVES SYNTEX LLC (US) 2003-06-18 EP disclosed
US-5719280-A REACTING AMINE SUBSTITUTED BENZOCYCLOALKANE WITH DIALKYLOXYACETALDEHYDE IN PRESENCE OF REDUCING AGENT OR CATALYTIC HYDROGENATION, TREATING WITH THIOCYANIC ACID SYNTEX (U.S.A.) INC. (US) 1998-02-17 US disclosed
EP-0757677-A1 BENZOCYCLOALKYLAZOLETHIONE DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1997-02-12 EP disclosed
US-5538988-A CARDIOVASCULAR DISORDERS AND DOPAMINE HYDROLASE ENZYME INHIBITORS SYNTEX (U.S.A.) INC. 1996-07-23 US disclosed
WO-1995029165-A2 BENZOCYCLOALKYLAZ0LETHIONE DERIVATIVES AS DOPAMIN BETA-HYDROXYLASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1995-11-02 WO disclosed