SCHEMBL6950820

SCHEMBL6950820

CCOc1ccc2[nH]c(CCCC(=O)N3CCCC(Cc4ccccc4)C3)cc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.47
HPGD P15428 6/20 0.47
KDM4E B2RXH2 5/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP2D6 P10635 1/20 0.47
HSD17B10 Q99714 3/20 0.47
TSHR P16473 2/20 0.47
BCHE P06276 3/20 0.44
MAOA P21397 3/20 0.44
ACHE P22303 3/20 0.44
MAOB P27338 3/20 0.44
MAPK1 P28482 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
LMNA P02545 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6949095 0.93 MEN1 (0.47) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL6954412 0.85 TACR3 (0.43) HPGDKDM4EMEN1KMT2AMAPK1
SCHEMBL6958058 0.85 MEN1 (0.55) HPGDKDM4EMEN1KMT2AMAPK1
SCHEMBL6953001 0.85 MEN1 (0.56) ALDH1A1KDM4EMEN1KMT2ATSHR
SCHEMBL6953902 0.83 DRD2 (0.44) HPGDKDM4EMEN1KMT2AMAPK1
SCHEMBL6959344 0.83 BCHE (0.46) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL6959388 0.83 TACR1 (0.51) ALDH1A1MEN1KMT2ABCHEACHE
SCHEMBL6958270 0.81 TACR1 (0.51) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL18782564 0.81 AKR1C3 (0.50) ALDH1A1HPGDSMN1; SMN2TACR3GRIN2D
SCHEMBL6956012 0.80 TACR3 (0.43) HPGDKDM4EMEN1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP disclosed
US-6333339-B1 CENTRAL SYSTEM DISORDERS, SCHIZOPHRENIA AND COGNITION ACTIVATORS MERCK PATENT GELLSCHAFT MIT BESCHRANKTER (DE) 2001-12-25 US disclosed
EP-0993458-A1 3-BENZYLPIPERIDINE MERCK PATENT GmbH (DE) 2000-04-19 EP disclosed
WO-1998057953-A1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 1998-12-23 WO disclosed