SCHEMBL6958270

SCHEMBL6958270

CCOc1ccc2c(CCCC(=O)N3CCCC(Cc4ccccc4)C3)c[nH]c2c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.51
TACR3 P29371 1/20 0.51
ALDH1A1 P00352 4/20 0.48
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
MC5R P33032 3/20 0.43
MC3R P41968 2/20 0.43
MC1R Q01726 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MAPK1 P28482 1/20 0.42
MAPT P10636 1/20 0.41
MC4R P32245 1/20 0.41
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
BCHE P06276 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6959388 0.94 TACR1 (0.51) TACR1TACR3ALDH1A1KMT2AMEN1
SCHEMBL6959582 0.92 TACR1 (0.52) TACR1TACR3ALDH1A1KMT2AMEN1
SCHEMBL6954843 0.86 TACR3 (0.55) TACR1TACR3ALDH1A1KMT2AMC5R
SCHEMBL6954934 0.86 TACR3 (0.55) TACR1TACR3ALDH1A1KMT2AMC5R
SCHEMBL6953209 0.85 TACR1 (0.52) TACR1TACR3ALDH1A1KMT2ABCHE
SCHEMBL6952765 0.84 TACR1 (0.52) TACR1TACR3ALDH1A1KMT2AMC5R
SCHEMBL6960163 0.83 CARM1 (0.45) KMT2AMEN1BCHE
SCHEMBL6949095 0.83 MEN1 (0.47) TACR3ALDH1A1KMT2AMEN1KDM4E
SCHEMBL6950820 0.81 ALDH1A1 (0.47) TACR3ALDH1A1KMT2AMEN1KDM4E
SCHEMBL6958451 0.81 TACR1 (0.55) TACR1TACR3ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP disclosed
US-6333339-B1 CENTRAL SYSTEM DISORDERS, SCHIZOPHRENIA AND COGNITION ACTIVATORS MERCK PATENT GELLSCHAFT MIT BESCHRANKTER (DE) 2001-12-25 US disclosed
EP-0993458-A1 3-BENZYLPIPERIDINE MERCK PATENT GmbH (DE) 2000-04-19 EP disclosed
WO-1998057953-A1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 1998-12-23 WO disclosed