SCHEMBL6954008

SCHEMBL6954008

COc1ccc2c(c1)C(CCN(C(C)=O)C(C)=O)CN2C(=O)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.47
ADORA3 P0DMS8 1/20 0.41
PRNP P04156 1/20 0.41
ALDH1A1 P00352 2/20 0.40
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TP53 P04637 1/20 0.40
ACHE P22303 2/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPKAPK2 P49137 1/20 0.38
P2RX4 Q99571 1/20 0.38
MMP9 P14780 3/20 0.38
MMP1 P03956 2/20 0.38
MMP3 P08254 2/20 0.38
MMP7 P09237 1/20 0.38
MMP13 P45452 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7131048 0.86 MTNR1A (0.52) HTR6ADORA3ALDH1A1NPSR1TP53
SCHEMBL9821509 0.70 GHSR (0.43)
SCHEMBL10347776 0.70 SRD5A1 (0.49) HTR6ALDH1A1NPSR1RAB9AMMP9
SCHEMBL9821560 0.69 GHSR (0.46)
SCHEMBL13947547 0.68 MAPT (0.47) HTR6ALDH1A1TP53NPC1RAB9A
SCHEMBL13964629 0.68 P2RY1 (0.48) HTR6ALDH1A1ACHEMMP9MMP1
SCHEMBL6943395 0.68 MTNR1A (0.61)
SCHEMBL15375250 0.68 NOTUM (0.58) ALDH1A1NPSR1PTGDR2NPC1RAB9A
SCHEMBL13947544 0.68 CACNA1G (0.50) HTR6ALDH1A1PTGDR2
SCHEMBL1310006 0.67 MTNR1A (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0851855-B9 ACYLATED DERIVATIVES OF MELATONIN AND ITS ANALOGUES, USEFUL AS MEDICAMENTS MACEF (FR) 2003-05-21 EP claimed
EP-0851855-B1 ACYLATED DERIVATIVES OF MELATONIN AND ITS ANALOGUES, USEFUL AS MEDICAMENTS MACEF (FR) 2002-06-05 EP claimed
US-6140372-A N-(2-(2-ACETYL-7-METHOXYNAPHTH-1-YL)ETHYL)ACETAMIDE; SEDATIVES; MELATONIN DISORDERS; DRUGS; COSMETICS; ANTIDEPRESSANTS; PSYCHIATRIC DISORDERS, E.G., STRESS, ANXIOLYTIC AGENTS, INSOMNIA, SCHIZOPHRENIA, PSYCHOSIS CEMAF AND LABORATORIES BESINS ISOVESCO S.A. (FR) 2000-10-31 US disclosed
US-6004991-A COMPOUNDS FOR COSMETICS WITH ENANTIOMORPHS CEMAF AND LABORATOIRES BESINS ISCOVESCO S.A. (FR) 1999-12-21 US disclosed