SCHEMBL6954009

SCHEMBL6954009

NOc1ccc(O)cc1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.43
TYR P14679 2/20 0.41
CES2 O00748 1/20 0.39
ALOX5 P09917 2/20 0.38
CA12 O43570 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA7 P43166 2/20 0.38
CA9 Q16790 2/20 0.38
CA14 Q9ULX7 2/20 0.38
TSHR P16473 1/20 0.38
SYNJ2 O15056 1/20 0.38
TTR P02766 1/20 0.38
CYP1A1 P04798 1/20 0.38
BCHE P06276 1/20 0.38
MMP2 P08253 1/20 0.38
PTPN1 P18031 1/20 0.38
PTGS1 P23219 1/20 0.38
CYP1B1 Q16678 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL278391 0.79 TTR (0.50) MAOBTYRCES2ALOX5CA12
SCHEMBL2198518 0.77 MAOB (0.44) MAOBTYRCES2ALOX5CA12
SCHEMBL68212 0.75 MAOB (0.67) MAOBALDH1A1CA1CA2TSHR
SCHEMBL29692356 0.75 MAOB (0.67) MAOBALDH1A1CA1CA2TSHR
SCHEMBL16182232 0.72 NPC1 (0.43) MAOBTYRALOX5ALDH1A1GFER
SCHEMBL5800656 0.72 TTR (0.61) CA12ALDH1A1CA1CA2CA7
SCHEMBL61461 0.72 ALDH1A1 (0.41) MAOBALDH1A1TSHRPTGS1
SCHEMBL14043320 0.72 BACE1 (0.33) MAOBALDH1A1ESR1IDO1
SCHEMBL13914988 0.71 MAOB (0.50) MAOBTYRCA12ALDH1A1CA1
SCHEMBL8819670 0.71 MAOB (0.40) MAOBTYRCES2ALOX5CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150247863-A1 DERIVATIVES OF 1,2-DIHYDRO-7-HYDROXYQUINOLINES CONTAINING FUSED RINGS Life Technologies Corporation 2015-09-03 US disclosed
US-20140356873-A1 Derivatives of 1,2-dihydro-7-hydroxyquinolines Containing Fused Rings LIFE TECHNOLOGIES CORP (US) 2014-12-04 US disclosed
US-8846925-B2 Derivatives of 1,2-dihydro-7-hydroxyquinolines containing fused rings Life Technologies Corporation (US) 2014-09-30 US disclosed
US-20120315661-A1 Derivatives of 1,2-dihydro-7-hydroxyquinolines Containing Fused Rings Life Technologies Corporation (US) 2012-12-13 US disclosed
US-8183375-B2 Derivatives of 1,2-dihydro-7-hydroxyquinolines containing fused rings Life Technologies Corporation (US) 2012-05-22 US disclosed
US-20110027800-A1 Derivatives of 1,2-dihydro-7-hydroxyquinolines Containing Fused Rings Life Technologies Corporation (US) 2011-02-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110027800-A1 Derivatives of 1,2-dihydro-7-hydroxyquinolines Containing Fused Rings CYP3A7, UGT1A7, UGT2B7 MAOB 1690/4885TYR 465/4885CES2 558/4885
US-20150247863-A1 DERIVATIVES OF 1,2-DIHYDRO-7-HYDROXYQUINOLINES CONTAINING FUSED RINGS CYP3A7, UGT1A7, UGT2B7 MAOB 1690/4885TYR 465/4885CES2 558/4885
US-20140356873-A1 Derivatives of 1,2-dihydro-7-hydroxyquinolines Containing Fused Rings CYP3A7, UGT1A7, UGT2B7 MAOB 1690/4885TYR 465/4885CES2 558/4885
US-20120315661-A1 Derivatives of 1,2-dihydro-7-hydroxyquinolines Containing Fused Rings CYP3A7, UGT1A7, UGT2B7 MAOB 1690/4885TYR 465/4885CES2 558/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.