SCHEMBL6954690

SCHEMBL6954690

C1=NC(Cc2ccc3ccccc3c2)CN1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 11/20 0.41
SLC6A4 P31645 11/20 0.41
SLC6A3 Q01959 11/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2A6 P11509 1/20 0.41
KCNH2 Q12809 2/20 0.40
CYP2D6 P10635 2/20 0.40
NFKB1 P19838 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR7 P34969 1/20 0.39
HTR2B P41595 1/20 0.39
HTR3A P46098 1/20 0.39
HTR4 Q13639 1/20 0.39
KDM1A O60341 2/20 0.38
MAOA P21397 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8084690 0.88 TBXA2R (0.43) SLC6A2SLC6A4SLC6A3CYP1A2KCNH2
Fumaric Acid SCHEMBL8084695 0.88 TBXA2R (0.43) SLC6A2SLC6A4SLC6A3CYP1A2KCNH2
SCHEMBL6957391 0.84 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3CYP1A2CYP2A6
SCHEMBL3441782 0.80 ADRA2A (0.42) TAAR1ADRA2A
SCHEMBL3441577 0.80 ADRA2A (0.42) TAAR1ADRA2A
SCHEMBL11821505 0.74 SLC6A4 (0.49) SLC6A2SLC6A4SLC6A3CYP1A2KCNH2
Fumaric Acid SCHEMBL8093564 0.72 ADRA2A (0.49) CYP1A2CYP2D6TAAR1CYP2C19ADRA2A
SCHEMBL3441406 0.72 CYP2D6 (0.51) CYP1A2CYP2D6TAAR1CYP2C9CYP2C19
SCHEMBL28262128 0.72 CYP1A2 (0.44) SLC6A2SLC6A4SLC6A3CYP1A2CYP2A6
SCHEMBL31392630 0.71 SLC6A4 (0.57) SLC6A2SLC6A4SLC6A3CYP1A2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1010693-B1 Imidazoline derivatives, preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-09-24 EP disclosed
EP-1010693-A1 Imidazoline derivatives, preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2000-06-21 EP disclosed