SCHEMBL6955084

SCHEMBL6955084

N=C(Nc1ccc(CCCN2CCCC2)cc1)c1cccs1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
LTA4H P09960 1/20 0.46
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPT P10636 3/20 0.42
LMNA P02545 1/20 0.42
FAAH O00519 1/20 0.42
HTT P42858 1/20 0.42
SIGMAR1 Q99720 3/20 0.42
OPRK1 P41145 1/20 0.41
POLB P06746 2/20 0.41
HRH1 P35367 1/20 0.40
L3MBTL3 Q96JM7 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GFER P55789 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6968037 0.99 ALDH1A1 (0.47) ALDH1A1KDM4EMEN1KMT2ALTA4H
SCHEMBL9039113 0.93 MEN1 (0.48) MEN1KMT2ANPC1TP53RAB9A
Hydrochloric Acid SCHEMBL9221658 0.92 MEN1 (0.47) ALDH1A1KDM4EMEN1KMT2ANPC1
Bromide SCHEMBL6967598 0.92 MEN1 (0.47) MEN1KMT2ANPC1TP53RAB9A
SCHEMBL8180687 0.92 MEN1 (0.47) ALDH1A1MEN1KMT2ANPC1TP53
Hydrochloric Acid SCHEMBL6962238 0.91 MEN1 (0.46) ALDH1A1KDM4EMEN1KMT2ANPC1
SCHEMBL6968869 0.87 DRD2 (0.47) ALDH1A1KDM4EMEN1KMT2ALTA4H
SCHEMBL6968837 0.85 SMN1; SMN2 (0.58) ALDH1A1KDM4EMEN1KMT2ANPC1
SCHEMBL9039593 0.84 SMN1; SMN2 (0.57) ALDH1A1KDM4EMEN1KMT2ANPC1
Bromide SCHEMBL8180586 0.84 SMN1; SMN2 (0.57) ALDH1A1KDM4EMEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed