SCHEMBL6955632

SCHEMBL6955632

Cc1nc(Nc2ccc(F)cc2)nc(N2CCc3ccc(OC(=O)COCc4ccccc4)cc3C2C)c1C

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.33
KCNH3 Q9ULD8 2/20 0.33
GRM5 P41594 1/20 0.33
DHFR P00374 3/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
KMT2A Q03164 1/20 0.32
PARP1 P09874 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
GHSR Q92847 1/20 0.31
CCNT1 O60563 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CDK9 P50750 1/20 0.31
CCNA1 P78396 1/20 0.31
CCKBR P32239 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957847 0.94 GRIN1 (0.36) EGFRKCNH3GRM5LMNATP53
SCHEMBL6969559 0.88 MEN1 (0.37) DHFRLMNATP53KMT2A
SCHEMBL6963615 0.87 KMT2A (0.35) EGFRLMNATP53KMT2A
SCHEMBL6970019 0.86 SMN1; SMN2 (0.37) EGFRKCNH3LMNATP53KMT2A
SCHEMBL6960659 0.85 POLB (0.38) EGFRKCNH3LMNAKMT2APARP1
SCHEMBL6966508 0.85 KMT2A (0.37) EGFRKCNH3TP53KMT2ACDK2
SCHEMBL6962677 0.85 SLC2A1 (0.40) EGFRKCNH3KMT2APARP1CDK2
Hydrochloric Acid SCHEMBL6966805 0.85 MC4R (0.34) KCNH3DHFRLMNATP53KMT2A
Hydrochloric Acid SCHEMBL6966802 0.85 MC4R (0.34) KCNH3DHFRLMNATP53KMT2A
SCHEMBL6955926 0.85 P2RX3 (0.34) EGFRLMNATP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015444-B1 PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP LTD (KR) 2003-05-28 EP claimed
EP-1015444-B1 PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP LTD (KR) 2003-05-28 EP disclosed
US-6352993-B1 ANTIULCER AGENTS YUHAN CORPORATION (KR) 2002-03-05 US disclosed