SCHEMBL6955656

SCHEMBL6955656

Cc1c(C(=O)CCn2ccnc2)sc2ccc(F)cc12

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 9/20 0.56
CYP19A1 P11511 2/20 0.46
PKM P14618 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
EGLN3 Q9H6Z9 1/20 0.40
TP53 P04637 1/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950423 0.87 TBXAS1 (0.56) TBXAS1PKMSMN1; SMN2TP53MAPK1
SCHEMBL1509582 0.84 TBXAS1 (0.53) TBXAS1CYP19A1PKMSMN1; SMN2EGLN3
SCHEMBL6964199 0.76 CXCR2 (0.42) TBXAS1PTGDR2
SCHEMBL6958299 0.76 CYP19A1 (0.46) TBXAS1CYP19A1
SCHEMBL14027515 0.72 TBXAS1 (0.54) TBXAS1CYP19A1
SCHEMBL11287283 0.72 TBXAS1 (1.00) TBXAS1
SCHEMBL6948774 0.72 POLB (0.60) TBXAS1CYP19A1EGLN3POLB
Hydrochloric Acid SCHEMBL7970769 0.72 TBXAS1 (0.42) TBXAS1CYP19A1PKMSMN1; SMN2KMT2A
SCHEMBL6955408 0.71 CYP19A1 (0.47) TBXAS1CYP19A1
SCHEMBL6955399 0.71 CYP19A1 (0.47) TBXAS1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0974584-B1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-15 EP disclosed
US-6420375-B1 ANTITUMOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-0974584-A1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-01-26 EP disclosed