SCHEMBL6958299

SCHEMBL6958299

Cc1c(C(O)CCn2ccnc2)sc2ccc(F)cc12

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.46
TBXAS1 P24557 6/20 0.43
QPCT Q16769 1/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6953884 0.87 ADRA2C (0.45) TBXAS1QPCT
SCHEMBL6955656 0.76 TBXAS1 (0.56) CYP19A1TBXAS1
SCHEMBL11635113 0.73 CYP19A1 (0.55) CYP19A1QPCTCYP11B1CYP11B2
SCHEMBL11633201 0.72 CYP19A1 (0.73) CYP19A1QPCTCYP11B1CYP11B2
SCHEMBL6955408 0.71 CYP19A1 (0.47) CYP19A1TBXAS1CYP11B1CYP11B2
SCHEMBL6955399 0.71 CYP19A1 (0.47) CYP19A1TBXAS1CYP11B1CYP11B2
SCHEMBL11392397 0.70 CYP19A1 (0.48) CYP19A1TBXAS1
SCHEMBL6963779 0.68 SIRT2 (0.39)
SCHEMBL12869982 0.67 CYP17A1 (0.44)
SCHEMBL11756428 0.67 CYP19A1 (0.53) CYP19A1QPCTCYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0974584-B1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-15 EP disclosed
US-6420375-B1 ANTITUMOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-0974584-A1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-01-26 EP disclosed