SCHEMBL6956030

SCHEMBL6956030

Fc1ccc2c(CCCCN3CCCC(Cc4ccccc4)C3)c[nH]c2c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.50
MPO P05164 2/20 0.50
SLC6A4 P31645 3/20 0.49
DRD4 P21917 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
HTR1D P28221 1/20 0.47
HTR1B P28222 1/20 0.47
ADRA1D P25100 2/20 0.46
CARM1 Q86X55 1/20 0.46
PRMT6 Q96LA8 1/20 0.46
HTR7 P34969 1/20 0.46
KCNH2 Q12809 1/20 0.46
DRD2 P14416 1/20 0.45
HTR2A P28223 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957729 0.93 MPO (0.61) HTR1AMPOSLC6A4HTR1DHTR1B
SCHEMBL6952634 0.93 MPO (0.61) HTR1AMPOSLC6A4HTR1DHTR1B
SCHEMBL6958552 0.93 MPO (0.61) HTR1AMPOSLC6A4HTR1DHTR1B
SCHEMBL6958541 0.89 SLC6A4 (0.49) HTR1ASLC6A4DRD4SIGMAR1HTR1D
SCHEMBL6950516 0.88 HTR1A (0.56) HTR1ASLC6A4HTR1DHTR1BCARM1
SCHEMBL6953004 0.87 MPO (0.63) HTR1AMPOSLC6A4
SCHEMBL6953432 0.86 SLC6A4 (0.52) HTR1ASLC6A4DRD2HTR2A
SCHEMBL6947219 0.86 HTR1A (0.52) HTR1ASLC6A4ADRA1DHTR2A
SCHEMBL6960163 0.85 CARM1 (0.45) HTR1ASLC6A4HTR1DHTR1BCARM1
SCHEMBL6951718 0.84 HTR1D (0.49) HTR1ASIGMAR1HTR1DHTR1BADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993458-B1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 2003-04-09 EP disclosed
US-6333339-B1 CENTRAL SYSTEM DISORDERS, SCHIZOPHRENIA AND COGNITION ACTIVATORS MERCK PATENT GELLSCHAFT MIT BESCHRANKTER (DE) 2001-12-25 US disclosed
EP-0993458-A1 3-BENZYLPIPERIDINE MERCK PATENT GmbH (DE) 2000-04-19 EP disclosed
WO-1998057953-A1 3-BENZYLPIPERIDINE MERCK PATENT GMBH (DE) 1998-12-23 WO disclosed