SCHEMBL6957825

SCHEMBL6957825

CC(=O)OCc1nc(C(C)C)c(Sc2cc(F)cc(F)c2)n1Cc1ccncc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 3/20 0.35
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
P2RX3 P56373 1/20 0.31
TP53 P04637 2/20 0.31
CYP19A1 P11511 1/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31
GRM5 P41594 1/20 0.30
CYP17A1 P05093 1/20 0.30
CYP21A2 P08686 1/20 0.30
CYP11B1 P15538 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6973130 0.92 ENPP2 (0.32) ENPP2MEN1KMT2ACYP19A1GRM5
SCHEMBL6973952 0.92 ENPP2 (0.36) ENPP2MEN1KMT2ACYP1A2CYP2C9
SCHEMBL6974519 0.92 ENPP2 (0.35) ENPP2MEN1KMT2AP2RX3TP53
SCHEMBL6969213 0.91 ENPP2 (0.35) ENPP2MEN1KMT2AP2RX3TP53
SCHEMBL6961984 0.90 ENPP2 (0.39) ENPP2MEN1KMT2AP2RX3TP53
SCHEMBL5852655 0.90 P2RX3 (0.33) ENPP2MEN1KMT2AP2RX3LMNA
SCHEMBL7079752 0.89 GRIN1 (0.37) ENPP2
SCHEMBL6975053 0.87 MEN1 (0.41) ENPP2MEN1KMT2ACYP1A2CYP2C9
SCHEMBL7083670 0.86 ENPP2 (0.33) ENPP2P2RX3
SCHEMBL6961792 0.86 ENPP2 (0.32) ENPP2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed