SCHEMBL6973952

SCHEMBL6973952

CC(=O)OCc1nc(C(C)C)c(Sc2cccc(F)c2)n1Cc1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.36
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
CYP2C9 P11712 4/20 0.34
CYP1A2 P05177 3/20 0.34
CYP2C19 P33261 3/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MAPT P10636 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
CYP3A4 P08684 3/20 0.33
CYP2D6 P10635 3/20 0.33
USP2 O75604 2/20 0.33
MIF P14174 1/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
SLC6A9 P48067 3/20 0.32
GRM2 Q14416 1/20 0.31
GRM5 P41594 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7086007 0.92 GRIN1 (0.33) ENPP2GRIN1GRIN2BCYP2C9CYP1A2
SCHEMBL6973183 0.92 ENPP2 (0.35) ENPP2GRIN1GRIN2BCYP2C9CYP1A2
SCHEMBL6957825 0.92 ENPP2 (0.35) ENPP2CYP2C9CYP1A2CYP2C19MEN1
SCHEMBL6975545 0.91 GRIN1 (0.34) ENPP2GRIN1GRIN2BCYP2C9CYP1A2
SCHEMBL6972338 0.91 GRIN1 (0.38) ENPP2GRIN1GRIN2BKMT2AMAPT
SCHEMBL6967603 0.91 ENPP2 (0.40) ENPP2GRIN1GRIN2BCYP2C9CYP1A2
SCHEMBL7081541 0.90 IDO1 (0.35) CYP2C9CYP1A2CYP2C19MEN1KMT2A
SCHEMBL6975053 0.89 MEN1 (0.41) ENPP2CYP2C9CYP1A2CYP2C19MEN1
SCHEMBL6967842 0.87 ENPP2 (0.33) ENPP2GRIN1GRIN2BLMNATP53
SCHEMBL6974491 0.87 MEN1 (0.37) CYP2C9CYP1A2CYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed