SCHEMBL6958225

SCHEMBL6958225

COc1ccc(Br)c(C=O)c1OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.50
SMN1; SMN2 Q16637 4/20 0.49
MAPT P10636 4/20 0.49
ALDH1A1 P00352 4/20 0.49
L3MBTL1 Q9Y468 3/20 0.49
LMNA P02545 1/20 0.49
HPGD P15428 1/20 0.49
BCHE P06276 6/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
HTR1A P08908 1/20 0.45
ADRA1D P25100 1/20 0.45
ADRA1A P35348 1/20 0.45
ADRA1B P35368 1/20 0.45
PTGER4 P35408 1/20 0.44
PTGER3 P43115 1/20 0.44
PTGER2 P43116 1/20 0.44
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3970773 0.86 BCHE (0.50) ERN1SMN1; SMN2MAPTL3MBTL1BCHE
SCHEMBL31562616 0.83 BCHE (0.48) ERN1SMN1; SMN2MAPTL3MBTL1LMNA
SCHEMBL31562251 0.81 LIPE (0.49) ERN1SMN1; SMN2MAPTL3MBTL1HPGD
SCHEMBL21823620 0.81 ERN1 (0.57) ERN1SMN1; SMN2MAPTALDH1A1L3MBTL1
SCHEMBL7746131 0.81 BCHE (0.48) ERN1SMN1; SMN2MAPTALDH1A1L3MBTL1
SCHEMBL28496730 0.79 PTPN1 (0.50) SMN1; SMN2MAPTALDH1A1L3MBTL1LMNA
SCHEMBL4883017 0.79 HTR1A (0.55) SMN1; SMN2MAPTALDH1A1L3MBTL1LMNA
SCHEMBL31663469 0.78 ERN1 (0.66) ERN1SMN1; SMN2MAPTALDH1A1L3MBTL1
SCHEMBL4374159 0.78 ERN1 (0.66) ERN1SMN1; SMN2MAPTALDH1A1L3MBTL1
SCHEMBL8032642 0.77 BCHE (0.50) ERN1L3MBTL1BCHEHTR1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250289789-A1 REVERSIBLE LYSINE COVALENT MODIFIERS OF CDK2 AND USES THEREOF TERREMOTO BIOSCIENCES, INC. 2025-09-18 US disclosed
WO-2025090658-A2 REVERSIBLE LYSINE COVALENT MODIFIERS OF CDK2 AND USES THEREOF TERREMOTO BIOSCIENCES, INC. (US) 2025-05-01 WO disclosed
US-20090215908-A1 TOLL LIKE RECEPTOR (TLR) SIGNALING ANTAGONIST RELIANCE LIFE SCIENCES PVT. LTD. (IN) 2009-08-27 US disclosed
US-20090048446-A1 Process For Producing Benzo[C]Phenanthridine Derivative NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2009-02-19 US disclosed
EP-0947514-B1 NOVEL PHENANETHRIDINIUM DERIVATIVES NIPPON KAYAKU KK (JP) 2003-02-12 EP disclosed
US-6187783-B1 ANTITUMOR AGENTS NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2001-02-13 US disclosed
EP-0947514-A1 NOVEL PHENANETHRIDINIUM DERIVATIVES NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1999-10-06 EP disclosed
EP-0487930-B1 Benzo[C]phenanthridinium derivatives NIPPON KAYAKU KK (JP) 1999-03-24 EP disclosed
US-5747502-A ANTITUMOR AGENTS, ANTIGROWTH AGENTS AND ANTICARCINOGENIC AGENTS NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1998-05-05 US disclosed
EP-0487930-A1 Process for preparing benzo[C]phenanthridinium derivatives, and novel compounds prepared by said process NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1992-06-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250289789-A1 REVERSIBLE LYSINE COVALENT MODIFIERS OF CDK2 AND USES THEREOF CDK2, CDK20, CDK1 ERN1 1389/4885SMN1; SMN2 2895/4885MAPT 3329/4885
US-20090215908-A1 TOLL LIKE RECEPTOR (TLR) SIGNALING ANTAGONIST TLR4, TLR5, TLR1 ERN1 2109/4885SMN1; SMN2 3760/4885MAPT 3117/4885
US-20090048446-A1 Process For Producing Benzo[C]Phenanthridine Derivative CBR1, CYP1A1, CBR3 ERN1 1109/4885SMN1; SMN2 2623/4885MAPT 4393/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.