SCHEMBL6958311

SCHEMBL6958311

N#CCc1c[c]cc(C#N)c1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ENPP2 Q13822 1/20 0.32
CYP2A6 P11509 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31
MMP3 P08254 1/20 0.31
FFAR1 O14842 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3335656 0.82 LOXL2 (0.35) CYP2A6LOXL2
SCHEMBL16959461 0.79 MEN1 (0.38) CYP2A6LOXL2MEN1KMT2A
SCHEMBL28049287 0.78 GRM5 (0.31) CYP2A6LOXL2
SCHEMBL28302773 0.78 LOXL2 (0.50) CYP2A6LOXL2
SCHEMBL16958767 0.78 GRM5 (0.33) CYP2A6LOXL2MEN1KMT2A
SCHEMBL458972 0.78 CYP2A6 (0.50) CYP2A6LOXL2MEN1KMT2A
SCHEMBL6965146 0.78 CYP2A6 (0.31) CYP2A6LOXL2MEN1KMT2A
SCHEMBL18301559 0.77 KDM4E (0.43) KDM4ETDP1ENPP2CYP2A6LOXL2
SCHEMBL501879 0.77 KDM4E (0.43) KDM4ETDP1ENPP2CYP2A6LOXL2
SCHEMBL16959862 0.76 TSHR (0.45) CYP2A6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1329160-A2 4-ACYLAMINOPYRAZOLE DERIVATIVES Sankyo Company, Limited (JP) 2003-07-23 EP disclosed