SCHEMBL6958381

SCHEMBL6958381

Fc1cccc(F)c1CCNC(=S)Nc1cnccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
RAB9A P51151 5/20 0.47
ALOX12 P18054 2/20 0.47
CDC7 O00311 1/20 0.46
AURKA O14965 1/20 0.46
PRKD3 O94806 1/20 0.46
MAP4K4 O95819 1/20 0.46
CDK1 P06493 1/20 0.46
CSF1R P07333 1/20 0.46
CDK2 P24941 1/20 0.46
MAPK1 P28482 1/20 0.46
FLT4 P35916 1/20 0.46
KDR P35968 1/20 0.46
CSNK1D P48730 1/20 0.46
CLK2 P49760 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
MAPK12 P53778 1/20 0.46
CSNK2A1 P68400 1/20 0.46
CDK5 Q00535 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6953648 0.84 ALDH1A1 (0.67) ALDH1A1RAB9AALOX12NPC1CYP1A2
SCHEMBL7082827 0.80 ALDH1A1 (0.72) ALDH1A1RAB9AALOX12MAPK1BCL6
SCHEMBL6905477 0.79 ALDH1A1 (0.67) ALDH1A1RAB9AALOX12NPC1CYP1A2
SCHEMBL29355134 0.79 RAB9A (0.67) ALDH1A1RAB9AALOX12NPC1CYP1A2
SCHEMBL30083706 0.79 LTC4S (0.56) ALDH1A1RAB9AALOX12NPC1HTT
SCHEMBL6953259 0.77 ALDH1A1 (0.60) ALDH1A1RAB9AALOX12MAPK1NPC1
SCHEMBL6961866 0.74 NPC1 (0.55) ALDH1A1RAB9AMAPK1NPC1CYP1A2
SCHEMBL6954353 0.74 RAB9A (0.42) ALDH1A1RAB9AALOX12NPC1CYP1A2
SCHEMBL6962081 0.74 POLB (0.58) ALDH1A1RAB9AALOX12NPC1CYP1A2
SCHEMBL6963213 0.73 ALDH1A1 (0.55) ALDH1A1RAB9AALOX12MAPK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0540143-B1 Compounds and methods for inhibition of HIV and related viruses MEDIVIR AB (SE) 2003-02-05 EP disclosed
US-5714503-A Compounds and methods for inhibition of HIV and related viruses MEDIVIR AB (SE) 1998-02-03 US disclosed
US-5658907-A THIOUREA VIRICIDES MEDIVIR A/B (SE) 1997-08-19 US disclosed
US-5593993-A VIRICIDES FOR HTLV TREATMENT OF AIDS MEDIVIR AB (SE) 1997-01-14 US disclosed
EP-0540143-A2 Compounds and methods for inhibition of HIV and related viruses Medivir Aktiebolag (SE) 1993-05-05 EP disclosed
WO-1993003022-A1 COMPOUNDS AND METHODS FOR INHIBITION OF HIV AND RELATED VIRUSES MEDIVIR AB (SE) 1993-02-18 WO disclosed