SCHEMBL6958498

SCHEMBL6958498

CC(C)c1ccccc1Sc1c(O)cc(-c2ccc(OCC(=O)O)cc2)oc1=O

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
AKR1C1 Q04828 1/20 0.40
THRB P10828 5/20 0.40
THRA P10827 4/20 0.40
MAPT P10636 3/20 0.38
KDM4E B2RXH2 2/20 0.38
PTPN7 P35236 1/20 0.38
POLB P06746 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961046 0.89 KDM4E (0.50) ALDH1A1HPGDTHRBMAPTKDM4E
SCHEMBL6965151 0.88 ABCB1 (0.45) MAPTL3MBTL1
SCHEMBL6954863 0.88 ABCB1 (0.39) SMN1; SMN2ALDH1A1HPGDMAPTKDM4E
SCHEMBL6966299 0.87 PPARD (0.41) THRBTHRAKDM4E
SCHEMBL6958195 0.86 ACHE (0.40) XDHMAPT
SCHEMBL6961094 0.86 NTRK1 (0.49) SMN1; SMN2ALDH1A1HPGDTHRBMAPT
SCHEMBL6961039 0.85 SMN1; SMN2 (0.46) XDHSMN1; SMN2ALDH1A1HPGDTHRB
SCHEMBL6958501 0.85 MAPT (0.39) SMN1; SMN2ALDH1A1HPGDMAPTKDM4E
SCHEMBL6952506 0.84 XDH (0.51) XDHSMN1; SMN2ALDH1A1HPGDAKR1C3
SCHEMBL6963494 0.83 PTGES (0.43) XDHSMN1; SMN2ALDH1A1HPGDTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729465-B1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & CO (US) 2003-01-22 EP disclosed
US-6005103-A TREATMENT OF BACTERIAL AND VIRAL INFECTIONS AND DISEASES, INCLUDING AIDS WARNER-LAMBERT COMPANY (US) 1999-12-21 US disclosed
EP-0729465-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
EP-0729466-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014013-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed
WO-1995014014-A2 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed