SCHEMBL6958838

SCHEMBL6958838

O=C([C@H]1CC[C@@H](CO)CC1)N(CCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.53
TACR1 P25103 16/20 0.46
ACHE P22303 1/20 0.45
SLC6A4 P31645 1/20 0.40
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6964535 0.90 HTT (0.52) HTTTACR1ACHESLC6A4CHRM5
SCHEMBL6964788 0.88 HTT (0.54) HTTTACR1ACHECHRM5CHRM1
SCHEMBL6965223 0.86 HTT (0.51) HTTTACR1ACHESLC6A4CHRM5
SCHEMBL6962588 0.83 HTT (0.49) HTTTACR1ACHE
SCHEMBL6957247 0.74 HTT (0.47) HTTTACR1
SCHEMBL4560442 0.69 HTT (0.63) HTTACHECHRM5CHRM1CHRM3
SCHEMBL5269885 0.65 HTT (0.47) HTTACHE
SCHEMBL1432538 0.65 GPBAR1 (0.50) TACR1SLC6A4CHRM5
SCHEMBL18930513 0.64 HTT (0.73) HTTACHESLC6A4
SCHEMBL9716647 0.64 HTT (0.74) HTTACHECHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286978-A1 CYCLOHEXYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 2003-03-05 EP disclosed
WO-2001087866-A1 CYCLOHEXYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 2001-11-22 WO disclosed