SCHEMBL6964535

SCHEMBL6964535

NC[C@H]1CC[C@H](C(=O)N(CCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c2ccccc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.52
ACHE P22303 1/20 0.44
TACR1 P25103 15/20 0.43
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA13 Q8N1Q1 1/20 0.38
CA14 Q9ULX7 1/20 0.38
SLC6A4 P31645 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958838 0.90 HTT (0.53) HTTACHETACR1CHRM5CHRM1
SCHEMBL6964788 0.89 HTT (0.54) HTTACHETACR1CHRM5CHRM1
SCHEMBL6965223 0.85 HTT (0.51) HTTACHETACR1CHRM5CHRM1
SCHEMBL6962588 0.82 HTT (0.49) HTTACHETACR1
SCHEMBL6957247 0.73 HTT (0.47) HTTTACR1
SCHEMBL4560442 0.68 HTT (0.63) HTTACHECHRM5CHRM1CHRM3
SCHEMBL5269885 0.65 HTT (0.47) HTTACHE
SCHEMBL18930513 0.64 HTT (0.73) HTTACHESLC6A4
SCHEMBL9716647 0.63 HTT (0.74) HTTACHECHRM3
SCHEMBL4969869 0.63 HTT (0.63) HTTACHECHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286978-A1 CYCLOHEXYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 2003-03-05 EP disclosed
WO-2001087866-A1 CYCLOHEXYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 2001-11-22 WO disclosed