SCHEMBL6965223

SCHEMBL6965223

O=C1CCC(C(=O)N(CCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c2ccccc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.51
TACR1 P25103 14/20 0.47
ACHE P22303 1/20 0.43
CHRM1 P11229 3/20 0.40
CHRM3 P20309 3/20 0.40
CHRM2 P08172 2/20 0.40
CHRM5 P08912 2/20 0.39
CHRM4 P08173 1/20 0.39
SLC6A4 P31645 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957247 0.89 HTT (0.47) HTTTACR1
SCHEMBL6964788 0.87 HTT (0.54) HTTTACR1ACHECHRM1CHRM3
SCHEMBL6958838 0.86 HTT (0.53) HTTTACR1ACHECHRM1CHRM3
SCHEMBL6964535 0.85 HTT (0.52) HTTTACR1ACHECHRM1CHRM3
SCHEMBL6962588 0.82 HTT (0.49) HTTTACR1ACHE
SCHEMBL4560442 0.70 HTT (0.63) HTTACHECHRM1CHRM3CHRM2
SCHEMBL6621794 0.66 TACR1 (0.49) TACR1
SCHEMBL2312935 0.65 LMNA (0.49) HTT
SCHEMBL5215277 0.64 TACR1 (0.40) TACR1
SCHEMBL2724136 0.63 HTT (0.71) HTTACHECHRM3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286978-A1 CYCLOHEXYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 2003-03-05 EP disclosed
WO-2001087866-A1 CYCLOHEXYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 2001-11-22 WO disclosed