SCHEMBL6959310

SCHEMBL6959310

COc1ccccc1COc1ccc(-c2cc(O)c(SCCc3ccccc3)c(=O)o2)cc1C

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PTGES O14684 3/20 0.40
FFAR4 Q5NUL3 3/20 0.38
CYP1A1 P04798 1/20 0.38
CYP1A2 P05177 1/20 0.38
ALOX5 P09917 1/20 0.38
RECQL P46063 1/20 0.38
TAAR1 Q96RJ0 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.37
CNR2 P34972 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
FFAR1 O14842 2/20 0.37
ANO1 Q5XXA6 1/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6964575 0.90 FFAR4 (0.44) ABCB1MEN1KMT2APTGESFFAR4
SCHEMBL6963656 0.88 CYP1A1 (0.44) ABCB1FFAR4CYP1A1CYP1A2FFAR1
SCHEMBL6959331 0.86 SYK (0.40) ABCB1PTGESFFAR4MRGPRX4MAOB
SCHEMBL6957747 0.85 CYP1A1 (0.50) ABCB1MEN1KMT2APTGESCYP1A1
SCHEMBL6963073 0.84 PPARD (0.43) MEN1KMT2AFFAR1
SCHEMBL6964221 0.84 HTR1A (0.41) FFAR4MRGPRX4MAOBBCHEACHE
SCHEMBL6959805 0.82 PTGS2 (0.46) MEN1KMT2APTGESALOX5MRGPRX4
SCHEMBL6964365 0.81 PTGES (0.47) ABCB1MEN1KMT2APTGESCYP1A1
SCHEMBL6961275 0.81 KDM4E (0.44) ABCB1MEN1KMT2APTGESALOX5
SCHEMBL6965249 0.81 HCAR2 (0.40) MEN1KMT2APTGESALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729465-B1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & CO (US) 2003-01-22 EP disclosed
US-6005103-A TREATMENT OF BACTERIAL AND VIRAL INFECTIONS AND DISEASES, INCLUDING AIDS WARNER-LAMBERT COMPANY (US) 1999-12-21 US disclosed
US-5808062-A AIDS THERAPY WARNER-LAMBERT COMPANY (US) 1998-09-15 US disclosed
EP-0729466-A1 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014014-A2 PYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed