SCHEMBL6960272

SCHEMBL6960272

CC(C)/C=N/N(C)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 12/20 0.44
KMT2A Q03164 12/20 0.44
MAPT P10636 11/20 0.44
TDP1 Q9NUW8 5/20 0.44
SMN1; SMN2 Q16637 7/20 0.41
RAB9A P51151 6/20 0.41
NPC1 O15118 5/20 0.41
ALDH1A1 P00352 5/20 0.41
MAPK1 P28482 4/20 0.41
HPGD P15428 1/20 0.41
POLB P06746 1/20 0.41
LMNA P02545 3/20 0.40
RELA Q04206 2/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
GAA P10253 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALOX12 P18054 2/20 0.37
HCRTR1 O43613 1/20 0.37
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21251507 0.81 MAPT (0.40) MEN1KMT2AMAPTTDP1SMN1; SMN2
SCHEMBL22473722 0.81 MEN1 (0.40) MEN1KMT2AMAPTTDP1SMN1; SMN2
SCHEMBL10671468 0.81 ALDH1A1 (0.43) MEN1KMT2AMAPTTDP1SMN1; SMN2
SCHEMBL12667811 0.76 MEN1 (0.47) MEN1KMT2AMAPTTDP1SMN1; SMN2
SCHEMBL9515353 0.76 MEN1 (0.47) MEN1KMT2AMAPTTDP1SMN1; SMN2
SCHEMBL6979719 0.76 MEN1 (0.47) MEN1KMT2AMAPTTDP1SMN1; SMN2
SCHEMBL13669995 0.75 MEN1 (0.41) MEN1KMT2AMAPTTDP1SMN1; SMN2
SCHEMBL22473651 0.72 MAPT (0.45) MEN1KMT2AMAPTTDP1SMN1; SMN2
SCHEMBL8494529 0.72 MAPT (0.57) MEN1KMT2AMAPTTDP1SMN1; SMN2
SCHEMBL8494526 0.72 MAPT (0.57) MEN1KMT2AMAPTTDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10787448-B2 Indolizino [3,2-C] quinoline-based fluorescent probe SEOUL NATIONAL UNIVERSITY R & DB FOUNDATION (KR) 2020-09-29 US disclosed
US-8349857-B2 Quinazoline derivatives having tyrosine kinase inhibitory activity SHIONOGI & CO., LTD. (JP) 2013-01-08 US disclosed
US-8202879-B2 Quinazoline derivatives having tyrosine kinase inhibitory activity SHIONOGI & CO., LTD. (JP) 2012-06-19 US disclosed
US-20120123114-A1 QUINAZOLINE DERIVATIVES HAVING TYROSINE KINASE INHIBITORY ACTIVITY SHIONOGI & CO., LTD. (JP) 2012-05-17 US disclosed
US-20090143414-A1 Quinazoline Derivatives Having Tyrosine Kinase Inhibitory Activity SHIONOGI & CO., LTD. (JP) 2009-06-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090143414-A1 Quinazoline Derivatives Having Tyrosine Kinase Inhibitory Activity ERBB2, EGFR, ABL1 MEN1 3302/4885KMT2A 1949/4885MAPT 4100/4885
US-20120123114-A1 QUINAZOLINE DERIVATIVES HAVING TYROSINE KINASE INHIBITORY ACTIVITY ERBB2, EGFR, ABL1 MEN1 3302/4885KMT2A 1949/4885MAPT 4100/4885
US-10787448-B2 Indolizino [3,2-C] quinoline-based fluorescent probe DNA2, IRF3, DDB1 MEN1 3101/4885KMT2A 3767/4885MAPT 1031/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.