SCHEMBL6960306

SCHEMBL6960306

CSc1ccc(COC2CN(OC(=O)OC(C)(C)C)CCC2c2ccc(OCCCOCc3cccs3)cc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
REN P00797 18/20 0.35
LTA4H P09960 1/20 0.32
EPHX2 P34913 1/20 0.32
GPR119 Q8TDV5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7079705 0.87 REN (0.42) REN
SCHEMBL6043886 0.85 REN (0.39) RENLTA4HEPHX2
SCHEMBL6958384 0.84 MEN1 (0.35) RENLTA4HEPHX2GPR119
SCHEMBL7080733 0.83 REN (0.45) REN
SCHEMBL7075890 0.83 REN (0.39) REN
SCHEMBL6956250 0.83 REN (0.47) REN
SCHEMBL7077432 0.83 REN (0.41) REN
SCHEMBL6961201 0.82 MAPT (0.45) RENGPR119
SCHEMBL6960968 0.81 GPR119 (0.40) RENGPR119
SCHEMBL7082632 0.81 REN (0.46) REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863875-B1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY HOFFMANN LA ROCHE (CH) 2003-06-04 EP disclosed
EP-0863875-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1998-09-16 EP disclosed
WO-1997009311-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1997-03-13 WO disclosed