SCHEMBL6961081

SCHEMBL6961081

C[C@@H]1Cc2cc(N3C[C@H](COS(C)(=O)=O)OC3=O)ccc2N1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.41
MAOA P21397 3/20 0.39
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39
LMNA P02545 1/20 0.39
PTGS1 P23219 1/20 0.39
CALML3 P27482 1/20 0.39
SDHA P31040 1/20 0.39
TNF P01375 8/20 0.39
NOD2 Q9HC29 8/20 0.39
NOD1 Q9Y239 7/20 0.39
GRM2 Q14416 4/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960931 0.85 MAOB (0.52) MAOBMAOATP53GAALMNA
SCHEMBL6968254 0.85 MAOB (0.52) MAOBMAOATP53GAALMNA
SCHEMBL6972540 0.84 F10 (0.44) MAOBMAOATP53GAALMNA
SCHEMBL6972140 0.81 MAOA (0.60) MAOBMAOALMNAPTGS1CALML3
SCHEMBL6214916 0.80 MAOB (0.40) MAOBMAOALMNAPTGS1CALML3
SCHEMBL6966689 0.79 MAOB (0.49) MAOBMAOALMNAPTGS1CALML3
SCHEMBL6961334 0.79 GRM2 (0.40) MAOBGRM2
SCHEMBL7485004 0.79 MAOB (0.57) MAOBMAOALMNAPTGS1CALML3
SCHEMBL7484998 0.79 MAOB (0.57) MAOBMAOALMNAPTGS1CALML3
SCHEMBL7597985 0.78 GRM2 (0.38) MAOBMAOAGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181288-B1 BICYCLIC OXAZOLIDINONES AS ANTIBACTERIAL AGENT UPJOHN CO (US) 2003-07-30 EP disclosed
US-20020143009-A1 Novel bicyclic oxazolidinones as antibacterial agents PHARMACIA & UPJOHN 2002-10-03 US disclosed
US-6387896-B1 GRAMNEGATIVE, GRAMPOSITVE BACTERIA PHARMACIA & UPJOHN CO. 2002-05-14 US disclosed
EP-1181288-A1 BICYCLIC OXAZOLIDINONES AS ANTIBACTERIAL AGENT PHARMACIA & UPJOHN COMPANY (US) 2002-02-27 EP disclosed
WO-2000073301-A1 BICYCLIC OXAZOLIDINONES AS ANTIBACTERIAL AGENT PHARMACIA & UPJOHN COMPANY (US) 2000-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020143009-A1 Novel bicyclic oxazolidinones as antibacterial agents OXA1L, MRPL21, RPS4Y1 MAOB 1600/4885MAOA 1716/4885TP53 4800/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.