SCHEMBL6961826

SCHEMBL6961826

NCCc1ccc(N=C(N)c2ccc[nH]2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.54
NOS3 P29474 4/20 0.54
NOS2 P35228 4/20 0.54
TAAR1 Q96RJ0 3/20 0.38
ADRA2A P08913 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HTR1A P08908 1/20 0.38
SLC6A2 P23975 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR3A P46098 1/20 0.38
BACE1 P56817 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
BLM P54132 1/20 0.37
KMT2A Q03164 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HTR2A P28223 2/20 0.36
CYP2A6 P11509 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6961986 0.74 KDM1A (0.50) ALDH1A1KMT2ASMN1; SMN2
SCHEMBL1428726 0.70
SCHEMBL1428727 0.70
SCHEMBL5378871 0.70 NOS1 (0.64) NOS1NOS3NOS2
SCHEMBL5378876 0.70 NOS1 (0.64) NOS1NOS3NOS2
SCHEMBL6961820 0.69 KDM1A (0.39) TAAR1ADRA2AKDM4EALDH1A1HTR1A
SCHEMBL8195295 0.67 CNR1 (0.49) KDM4EALDH1A1SLC6A2L3MBTL1KMT2A
SCHEMBL1972667 0.67
SCHEMBL27447143 0.67 NOS3 (0.54) NOS1NOS3NOS2TAAR1ADRA2A
Hydrochloric Acid SCHEMBL9213909 0.66 NOS3 (0.55) NOS1NOS3NOS2TAAR1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO claimed
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed