SCHEMBL6961986

SCHEMBL6961986

NC(=Nc1ccc(CCCC(=O)Nc2ccccc2)cc1)c1ccc[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.50
HDAC1 Q13547 3/20 0.48
HDAC2 Q92769 3/20 0.48
HDAC3 O15379 2/20 0.48
HDAC4 P56524 2/20 0.48
HDAC7 Q8WUI4 2/20 0.48
HDAC10 Q969S8 2/20 0.48
HDAC11 Q96DB2 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
HDAC9 Q9UKV0 2/20 0.48
HDAC5 Q9UQL6 2/20 0.48
TRPV1 Q8NER1 1/20 0.48
MAPT P10636 3/20 0.45
HTT P42858 1/20 0.45
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
ALDH1A1 P00352 1/20 0.45
ALOX15 P16050 1/20 0.45
NFKB1 P19838 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9037006 0.87 KDM1A (0.50) KDM1AHDAC1HDAC2HDAC3HDAC4
SCHEMBL6961976 0.80 TRPV1 (0.55) KDM1AHDAC1HDAC2HDAC3HDAC4
SCHEMBL6962660 0.78 NOS1 (0.59) KDM1AHDAC1HDAC2HDAC3HDAC4
SCHEMBL6970057 0.77 KDM1A (0.48) KDM1AHDAC1HDAC2HDAC3HDAC4
SCHEMBL6970018 0.76 KDM1A (0.47) KDM1AHDAC1HDAC2HDAC3HDAC4
SCHEMBL8394220 0.75 KDM1A (0.51) KDM1AHDAC1HDAC2HDAC3HDAC4
SCHEMBL6961826 0.74 NOS1 (0.54) ALDH1A1SMN1; SMN2KMT2A
SCHEMBL8012743 0.74 TRPV1 (0.81) KDM1AHDAC1HDAC2HDAC3HDAC4
SCHEMBL6961827 0.73 KDM1A (0.68) KDM1AHDAC1HDAC2HDAC3HDAC4
Hydrochloric Acid SCHEMBL8392010 0.72 KDM1A (0.66) KDM1AHDAC1HDAC2HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO claimed
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed