SCHEMBL6962306

SCHEMBL6962306

Cn1nnc(-c2ccc3[nH]cc(C4=CCNCC4)c3c2)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.55
ALDH1A1 P00352 3/20 0.55
HTR2C P28335 3/20 0.55
HSD17B10 Q99714 3/20 0.55
HTR1D P28221 3/20 0.55
MAPT P10636 2/20 0.55
HTR6 P50406 2/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
MAPK1 P28482 1/20 0.55
BRCA1 P38398 1/20 0.55
JAK2 O60674 1/20 0.53
PRKD3 O94806 1/20 0.53
MARK3 P27448 1/20 0.53
PRKCI P41743 1/20 0.53
PRKCD Q05655 1/20 0.53
CAMK2B Q13554 1/20 0.53
CAMK2G Q13555 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7392593 0.76 JAK2 (0.69) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL6954562 0.75 DRD2 (0.56) HTR2CHTR6DRD2HTR1B
SCHEMBL6960967 0.75 DRD2 (0.48) HTR2CHTR6DRD2HTR1B
SCHEMBL6631651 0.74 KDM4E (0.70) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL9093496 0.73 ALDH1A1 (0.56) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL9094194 0.72 HTR6 (0.55) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL9094655 0.72 KDM4E (0.55) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL9094872 0.72 JAK2 (0.55) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL2778860 0.71 HTR6 (0.67) KDM4EALDH1A1HTR2CHSD17B10HTR1D
SCHEMBL3836149 0.71 HTR6 (0.67) KDM4EALDH1A1HTR2CHSD17B10HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602889-B1 5-heteroaryl substituted indoles H. LUNDBECK A.S. (DK) 2003-08-05 US disclosed
EP-1068198-B1 5-HETEROARYL SUBSTITUTED INDOLES LUNDBECK & CO AS H (DK) 2003-05-28 EP disclosed