SCHEMBL696285

SCHEMBL696285

Nc1nc(-c2ccccc2)cc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.56
ADORA2A P29274 4/20 0.55
ADORA1 P30542 4/20 0.55
CYP1A1 P04798 1/20 0.49
CYP1B1 Q16678 1/20 0.49
MAPT P10636 3/20 0.48
MEN1 O00255 3/20 0.48
ALDH1A1 P00352 3/20 0.48
HPGD P15428 3/20 0.48
KMT2A Q03164 3/20 0.48
ADORA3 P0DMS8 1/20 0.47
KDM4E B2RXH2 2/20 0.47
HSP90AA1 P07900 1/20 0.47
HSP90AB1 P08238 1/20 0.47
IDO1 P14902 1/20 0.46
TDO2 P48775 1/20 0.46
LMNA P02545 1/20 0.46
AGTR1 P30556 1/20 0.46
SMARCA2 P51531 1/20 0.46
SMARCA4 P51532 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL28322407 0.86 SYK (0.52) ACHEADORA2AADORA1MAPTALDH1A1
SCHEMBL7978412 0.85 ALDH1A1 (0.57) ACHEMAPTMEN1ALDH1A1HPGD
SCHEMBL509835 0.85 ADORA2A (0.52) ACHEADORA2AADORA1MEN1ALDH1A1
SCHEMBL5529985 0.83 ADORA2A (0.47) ACHEADORA2AMAPTMEN1ALDH1A1
SCHEMBL509836 0.83 CYP11B1 (0.57) ADORA2AMAPTMEN1ALDH1A1HPGD
SCHEMBL508694 0.83 MAP4K4 (0.54) ADORA2AADORA1BACE1
SCHEMBL6634946 0.80 KDM4E (0.51) ACHEADORA2AADORA1MAPTMEN1
SCHEMBL11375277 0.80 KDM4E (0.50) ACHEADORA2AADORA1MAPTMEN1
SCHEMBL29177933 0.80 ACHE (0.52) ACHEADORA2AADORA1CYP1A1CYP1B1
SCHEMBL509600 0.79 ADORA2A (0.53) ADORA2AADORA1ADORA3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2935293-B1 IRIDIUM COMPLEXES AND THEIR USE IN ELECTRONIC DEVICES, ESPECIALLY ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2019-08-21 EP disclosed
CN-107428692-A Substituted monoazanaphthalene derivatives and polyazanaphthalene derivatives and use thereof 巴斯利尔药物国际股份公司 2017-12-01 CN disclosed
US-20150318498-A1 Metal Complexes MERCK PATENT GMBH (DE) 2015-11-05 US disclosed
US-20150318498-A1 Metal Complexes MERCK PATENT GMBH (DE) 2015-11-05 US disclosed
WO-2014094962-A2 METAL COMPLEXES MERCK PATENT GMBH (DE) 2014-06-26 WO disclosed
EP-2423196-A1 5, 6 or 7-substituted-3-phenylisoquinolinamine derivatives and therapeutic use thereof Rexahn Pharmaceuticals, Inc. (US) 2012-02-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150318498-A1 Metal Complexes SOD1, AP1M1, AP3M1 ACHE 2257/4885ADORA2A 4811/4885ADORA1 4851/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.