SCHEMBL6962946

SCHEMBL6962946

Nc1ccccc1CC(=O)NCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
LMNA P02545 1/20 0.58
HDAC3 O15379 2/20 0.58
HDAC4 P56524 2/20 0.58
HDAC1 Q13547 2/20 0.58
HDAC7 Q8WUI4 2/20 0.58
HDAC2 Q92769 2/20 0.58
HDAC10 Q969S8 2/20 0.58
HDAC11 Q96DB2 2/20 0.58
HDAC8 Q9BY41 2/20 0.58
HDAC6 Q9UBN7 2/20 0.58
HDAC9 Q9UKV0 2/20 0.58
HDAC5 Q9UQL6 2/20 0.58
RAB9A P51151 3/20 0.57
GAA P10253 2/20 0.57
MAPT P10636 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
CA12 O43570 2/20 0.55
CA1 P00915 2/20 0.55
CA2 P00918 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5161911 0.84 ALDH1A1 (0.53) ALDH1A1LMNAHDAC3HDAC4HDAC1
SCHEMBL5162641 0.83 ALDH1A1 (0.51) ALDH1A1LMNAHDAC3HDAC4HDAC1
SCHEMBL392625 0.81 ALDH1A1 (0.82) ALDH1A1LMNAHDAC3HDAC4HDAC1
SCHEMBL25046059 0.79 ALDH1A1 (0.65) ALDH1A1LMNARAB9AGAAMAPT
SCHEMBL28992287 0.79 ERCC1 (0.68) ALDH1A1LMNARAB9AGAAMAPT
SCHEMBL6962953 0.79 ALDH1A1 (0.73) ALDH1A1LMNAHDAC3HDAC4HDAC1
SCHEMBL1568340 0.79 ALDH1A1 (0.70) ALDH1A1LMNARAB9AGAAMAPT
SCHEMBL4717861 0.79 CA12 (0.71) ALDH1A1LMNAHDAC3HDAC4HDAC1
SCHEMBL14278969 0.79 TAAR1 (0.42) ALDH1A1HDAC3HDAC4HDAC1HDAC7
SCHEMBL27536085 0.78 FDPS (0.44) ALDH1A1HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed