SCHEMBL6963117

SCHEMBL6963117

O=C(CCCn1ccnc1)c1ccc2ccccc2c1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 5/20 0.64
HDAC1 Q13547 2/20 0.50
HDAC8 Q9BY41 1/20 0.50
CYP19A1 P11511 1/20 0.50
KDM4E B2RXH2 2/20 0.49
HPGD P15428 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ALDH1A1 P00352 1/20 0.48
SOD1 P00441 1/20 0.48
NAMPT P43490 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11253238 0.92 TBXAS1 (0.56) TBXAS1CYP19A1KDM4EHPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL11252177 0.91 TBXAS1 (0.55) TBXAS1CYP19A1KDM4EHPGDSMN1; SMN2
Nafimidone SCHEMBL1817018 0.84 ALPG (0.66) TBXAS1CYP19A1
SCHEMBL6949512 0.84 TBXAS1 (0.89) TBXAS1CYP19A1
Nafimidone SCHEMBL29861032 0.83 ALPG (0.67) TBXAS1CYP19A1
Nafimidone SCHEMBL412582 0.83 ALPG (0.67) TBXAS1CYP19A1
Hydrochloric Acid SCHEMBL11259498 0.82 TBXAS1 (0.86) TBXAS1CYP19A1
Nafimidone SCHEMBL11356554 0.82 ALPG (0.63) TBXAS1CYP19A1
SCHEMBL11152430 0.81 TBXAS1 (0.70) TBXAS1CYP19A1ALDH1A1
SCHEMBL2436231 0.81 TBXAS1 (0.59) TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0974584-B1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-15 EP disclosed
US-6420375-B1 ANTITUMOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
CN-1251577-A Fused ring compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-04-26 CN disclosed
EP-0974584-A1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-01-26 EP disclosed