SCHEMBL6963390

SCHEMBL6963390

O=C(N(Cc1ccccc1)Cc1cccc([N+](=O)[O-])c1)C(F)(F)F

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.59
LMNA P02545 3/20 0.59
CYP1A2 P05177 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
CRHBP P24387 1/20 0.53
CRHR2 Q13324 1/20 0.53
PKM P14618 2/20 0.53
HTT P42858 3/20 0.48
KDM4E B2RXH2 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
TSHR P16473 1/20 0.47
CTSB P07858 1/20 0.46
FAAH O00519 1/20 0.46
MGLL Q99685 1/20 0.46
PYCR1 P32322 1/20 0.46
MAPK1 P28482 1/20 0.46
RAB9A P51151 3/20 0.46
NPC1 O15118 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16366561 0.90 ALDH1A1 (0.50) ALDH1A1LMNACYP1A2CYP2D6CYP2C9
SCHEMBL6957148 0.88 CRHBP (0.65) ALDH1A1LMNACYP1A2CYP2C19CRHBP
SCHEMBL3441973 0.85 ALDH1A1 (0.48) ALDH1A1LMNACYP1A2CYP2D6CYP2C9
SCHEMBL6967315 0.85 KCNH2 (0.58) ALDH1A1LMNACYP1A2CYP2D6CYP2C9
SCHEMBL3442513 0.85 ALDH1A1 (0.46) ALDH1A1LMNACYP1A2CYP2D6CYP2C9
SCHEMBL3441758 0.83 PYCR1 (0.53) ALDH1A1LMNACYP1A2CYP2D6CYP2C9
SCHEMBL3861529 0.81 CYP1A2 (0.44) ALDH1A1LMNACYP1A2CYP2D6CYP2C9
SCHEMBL16373478 0.81 CES1 (0.52) ALDH1A1LMNACYP1A2CYP2C9CYP2C19
SCHEMBL25376679 0.80 ALDH1A1 (0.60) ALDH1A1LMNACYP1A2CYP2D6CYP2C9
SCHEMBL15265399 0.80 ALDH1A1 (0.64) ALDH1A1LMNACYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0713483-B1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRAZENECA AB (SE) 2003-01-15 EP disclosed
US-6030985-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 2000-02-29 US disclosed
US-5807885-A Amidine derivatives with nitric oxide synthetase activities ASTRA AKTIEBOLAG (SE) 1998-09-15 US disclosed
WO-1995005363-A1 AMIDINE DERIVATIVES WITH NITRIC OXIDE SYNTHETASE ACTIVITIES ASTRA AKTIEBOLAG (SE) 1995-02-23 WO disclosed