SCHEMBL6963904

SCHEMBL6963904

NC(=O)c1ccc(S(=O)(=O)c2cccc3cnccc23)c([N+](=O)[O-])c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.47
MEN1 O00255 6/20 0.44
KMT2A Q03164 6/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
ALDH1A1 P00352 3/20 0.43
GAA P10253 1/20 0.43
PARP1 P09874 1/20 0.41
MELK Q14680 2/20 0.41
MAPK1 P28482 1/20 0.41
CAMKK2 Q96RR4 1/20 0.41
HIPK2 Q9H2X6 1/20 0.41
LMNA P02545 3/20 0.41
HTT P42858 2/20 0.41
HPGD P15428 1/20 0.41
PRKD3 O94806 3/20 0.41
PRKCG P05129 3/20 0.41
PRKCB P05771 3/20 0.41
CYP3A4 P08684 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6965038 0.85 CYP3A4 (0.44) MEN1KMT2AKDM4ETDP1ALDH1A1
SCHEMBL6958223 0.79 P2RX7 (0.42) MEN1KMT2AMAPTKDM4ETDP1
SCHEMBL6977470 0.77 CYP3A4 (0.44) POLBMEN1KMT2AKDM4ETDP1
SCHEMBL6975024 0.76 CYP19A1 (0.44) MEN1KMT2AKDM4EALDH1A1MELK
SCHEMBL6963085 0.76 CYP3A4 (0.44) MEN1KMT2AKDM4ETDP1MELK
SCHEMBL6977825 0.76 KDM4E (0.43) MEN1KMT2AKDM4EMELKMAPK1
SCHEMBL6966488 0.76 MEN1 (0.44) MEN1KMT2AKDM4EALDH1A1MAPK1
SCHEMBL6962005 0.75 NPY1R (0.43) MEN1KMT2AKDM4EMELKMAPK1
SCHEMBL6976355 0.75 NPY1R (0.43) MEN1KMT2AMAPTKDM4ETDP1
SCHEMBL6970886 0.75 PRKD3 (0.43) MEN1KMT2AMAPTKDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed