SCHEMBL6977825

SCHEMBL6977825

O=[N+]([O-])c1ccc(S(=O)(=O)c2cccc3cnccc23)cc1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
MAPKAPK2 P49137 1/20 0.43
HTR6 P50406 1/20 0.43
P2RX7 Q99572 2/20 0.42
NAMPT P43490 2/20 0.41
PRKD3 O94806 4/20 0.41
PRKCG P05129 4/20 0.41
PRKCB P05771 4/20 0.41
CYP3A4 P08684 4/20 0.41
PRKCA P17252 4/20 0.41
PRKCH P24723 4/20 0.41
PRKCI P41743 4/20 0.41
PRKCE Q02156 4/20 0.41
PRKCQ Q04759 4/20 0.41
PRKCZ Q05513 4/20 0.41
PRKCD Q05655 4/20 0.41
PRKD1 Q15139 4/20 0.41
MEN1 O00255 3/20 0.41
CYP2D6 P10635 3/20 0.41
PRKACA P17612 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6963085 0.86 CYP3A4 (0.44) KDM4EHTR6P2RX7PRKD3PRKCG
SCHEMBL6977470 0.85 CYP3A4 (0.44) KDM4EHTR6P2RX7PRKD3PRKCG
SCHEMBL6961086 0.82 CYP3A4 (0.47) KDM4EMAPKAPK2HTR6P2RX7NAMPT
SCHEMBL6961874 0.80 P2RX7 (0.52) KDM4EHTR6P2RX7PRKD3PRKCG
SCHEMBL6966488 0.79 MEN1 (0.44) KDM4EP2RX7PRKD3PRKCGPRKCB
SCHEMBL6962809 0.78 HTR6 (0.44) KDM4EMAPKAPK2HTR6P2RX7NAMPT
SCHEMBL6965038 0.78 CYP3A4 (0.44) KDM4EHTR6P2RX7PRKD3PRKCG
SCHEMBL6971028 0.77 CYP3A4 (0.44) KDM4EP2RX7PRKD3PRKCGPRKCB
SCHEMBL6963904 0.76 POLB (0.47) KDM4EP2RX7PRKD3PRKCGPRKCB
SCHEMBL22005940 0.76 TXNRD1 (0.50) KDM4ECYP3A4MEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed