SCHEMBL6964345

SCHEMBL6964345

CCOC(=O)C=Cc1cc2ccc(F)cc2s1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.43
TDO2 P48775 1/20 0.43
TTR P02766 1/20 0.43
DPP4 P27487 1/20 0.43
PTPN1 P18031 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
MAPT P10636 3/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 2/20 0.41
NPC1 O15118 1/20 0.41
ALPL P05186 1/20 0.41
HPGD P15428 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6964344 1.00 IDO1 (0.43) IDO1TDO2TTRDPP4PTPN1
SCHEMBL14016232 0.84 ESR1 (0.43) TTRDPP4CA12CA1CA2
SCHEMBL6965215 0.83 CYP2A6 (0.47) TTRDPP4CA12CA1CA2
SCHEMBL6965217 0.83 CYP2A6 (0.47) TTRDPP4CA12CA1CA2
SCHEMBL9540314 0.78 FDPS (0.50) TTRDPP4CYP3A4HSD17B1HSD17B2
SCHEMBL29427194 0.77 TP53 (0.50) MAPTALDH1A1NPC1HPGDRAB9A
SCHEMBL29709927 0.77 TTR (0.43) TTRDPP4CA12CA1CA2
SCHEMBL6965431 0.77 MAPT (0.44) TTRDPP4PTPN1CA12CA1
SCHEMBL6965434 0.77 MAPT (0.44) TTRDPP4PTPN1CA12CA1
SCHEMBL2325697 0.76 CYP3A4 (0.51) IDO1TDO2TTRDPP4CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0974584-B1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-15 EP disclosed
US-6420375-B1 ANTITUMOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed
EP-0974584-A1 FUSED RING COMPOUNDS, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-01-26 EP disclosed