SCHEMBL6965245

SCHEMBL6965245

Nc1cc(Sc2cccc3cnccc23)c(Br)cc1[N+](=O)[O-]

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAPT P10636 5/20 0.41
TDP1 Q9NUW8 4/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
GAA P10253 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MAPK1 P28482 1/20 0.41
PDE7A Q13946 8/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 3/20 0.38
HTT P42858 2/20 0.38
CTSB P07858 1/20 0.38
PSMD14 O00487 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972315 0.91 LMNA (0.46) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6958271 0.89 LMNA (0.42) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6965142 0.87 PDE7A (0.47) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6963335 0.86 LMNA (0.46) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6958268 0.84 LMNA (0.42) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6966276 0.84 MAPT (0.42) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6966094 0.82 LMNA (0.43) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6968103 0.81 MAPT (0.48) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6976355 0.77 NPY1R (0.43) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8357964 0.76 SLC6A2 (0.49) LMNACYP3A4MAPTTDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed